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Design, synthesis and biological evaluation of novel aminopyrazole- and 7-azaindole-based Nek1 inhibitors and their effects on zebrafish kidney development.
Pilakowski, Johannes; Baumann, Georg; Shih, Yung-Hsin; Meckel, Tobias; Schmidt, Boris.
Afiliação
  • Pilakowski J; Clemens-Schöpf-Institute of Organic Chemistry and Biochemistry, Technische Universität Darmstadt, 64287 Darmstadt, Germany.
  • Baumann G; Clemens-Schöpf-Institute of Organic Chemistry and Biochemistry, Technische Universität Darmstadt, 64287 Darmstadt, Germany.
  • Shih YH; Clemens-Schöpf-Institute of Organic Chemistry and Biochemistry, Technische Universität Darmstadt, 64287 Darmstadt, Germany.
  • Meckel T; Ernst-Berl-Institute, Group of Macromolecular Chemistry and Paper Chemistry, Technische Universität Darmstadt, 64287 Darmstadt, Germany.
  • Schmidt B; Clemens-Schöpf-Institute of Organic Chemistry and Biochemistry, Technische Universität Darmstadt, 64287 Darmstadt, Germany. Electronic address: schmidt_boris@mac.com.
Bioorg Med Chem Lett ; 53: 128418, 2021 12 01.
Article em En | MEDLINE | ID: mdl-34715306

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirazóis / Desenho de Fármacos / Inibidores de Proteínas Quinases / Quinase 1 Relacionada a NIMA / Indóis / Rim Limite: Animals Idioma: En Revista: Bioorg Med Chem Lett Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirazóis / Desenho de Fármacos / Inibidores de Proteínas Quinases / Quinase 1 Relacionada a NIMA / Indóis / Rim Limite: Animals Idioma: En Revista: Bioorg Med Chem Lett Ano de publicação: 2021 Tipo de documento: Article