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The discovery of a novel series of potential ERRα inverse agonists based on p-nitrobenzenesulfonamide template for triple-negative breast cancer in vivo.
Gao, Zhipei; Wang, Tianxiao; Li, Rui; Du, Yongli; Lv, Han; Zhang, Liudi; Chen, Haifei; Shi, Xiaojin; Li, Qunyi; Shen, Jingkang.
Afiliação
  • Gao Z; School of Chemistry and Chemical Engineering, Qilu University of Technology (Shandong Academy of Sciences), Jinan, P. R. China.
  • Wang T; Department of Pharmacy, Huashan Hospital, Fudan University, Shanghai, P. R. China.
  • Li R; School of Chemistry and Chemical Engineering, Qilu University of Technology (Shandong Academy of Sciences), Jinan, P. R. China.
  • Du Y; School of Chemistry and Chemical Engineering, Qilu University of Technology (Shandong Academy of Sciences), Jinan, P. R. China.
  • Lv H; School of Chemistry and Chemical Engineering, Qilu University of Technology (Shandong Academy of Sciences), Jinan, P. R. China.
  • Zhang L; Department of Pharmacy, Huashan Hospital, Fudan University, Shanghai, P. R. China.
  • Chen H; Department of Pharmacy, Huashan Hospital, Fudan University, Shanghai, P. R. China.
  • Shi X; Department of Pharmacy, Huashan Hospital, Fudan University, Shanghai, P. R. China.
  • Li Q; Department of Pharmacy, Huashan Hospital, Fudan University, Shanghai, P. R. China.
  • Shen J; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, P. R. China.
J Enzyme Inhib Med Chem ; 37(1): 125-134, 2022 Dec.
Article em En | MEDLINE | ID: mdl-34894977

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Sulfonamidas / Receptores de Estrogênio / Descoberta de Drogas / Neoplasias de Mama Triplo Negativas / Antineoplásicos / Nitrobenzenos Limite: Female / Humans Idioma: En Revista: J Enzyme Inhib Med Chem Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Sulfonamidas / Receptores de Estrogênio / Descoberta de Drogas / Neoplasias de Mama Triplo Negativas / Antineoplásicos / Nitrobenzenos Limite: Female / Humans Idioma: En Revista: J Enzyme Inhib Med Chem Ano de publicação: 2022 Tipo de documento: Article