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Design, synthesis, and behavioral evaluation of dual-acting compounds as phosphodiesterase type 10A (PDE10A) inhibitors and serotonin ligands targeting neuropsychiatric symptoms in dementia.
Zagórska, Agnieszka; Bucki, Adam; Partyka, Anna; Jastrzebska-Wiesek, Magdalena; Siwek, Agata; Gluch-Lutwin, Monika; Mordyl, Barbara; Jaromin, Anna; Walczak, Maria; Wesolowska, Anna; Kolaczkowski, Marcin.
Afiliação
  • Zagórska A; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland. Electronic address: agnieszka.zagorska@uj.edu.pl.
  • Bucki A; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
  • Partyka A; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
  • Jastrzebska-Wiesek M; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
  • Siwek A; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
  • Gluch-Lutwin M; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
  • Mordyl B; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
  • Jaromin A; Department of Lipids and Liposomes, Faculty of Biotechnology, University of Wroclaw, 14a Joliot-Curie Street, 50-383, Wroclaw, Poland.
  • Walczak M; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
  • Wesolowska A; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
  • Kolaczkowski M; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
Eur J Med Chem ; 233: 114218, 2022 Apr 05.
Article em En | MEDLINE | ID: mdl-35248836

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antipsicóticos / Demência Tipo de estudo: Diagnostic_studies Limite: Animals / Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antipsicóticos / Demência Tipo de estudo: Diagnostic_studies Limite: Animals / Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2022 Tipo de documento: Article