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GNE-064: A Potent, Selective, and Orally Bioavailable Chemical Probe for the Bromodomains of SMARCA2 and SMARCA4 and the Fifth Bromodomain of PBRM1.
Taylor, Alexander M; Bailey, Chris; Belmont, Lisa D; Campbell, Robert; Cantone, Nico; Côté, Alexandre; Crawford, Terry D; Cummings, Richard; DeMent, Kevin; Duplessis, Martin; Flynn, Megan; Good, Andrew C; Huang, Hon-Ren; Joshi, Shivangi; Leblanc, Yves; Murray, Jeremy; Nasveschuk, Christopher G; Neiss, Adrianne; Poy, Florence; Romero, F Anthony; Sandy, Peter; Tang, Yong; Tsui, Vickie; Zawadzke, Laura; Sims, Robert J; Audia, James E; Bellon, Steven F; Magnuson, Steven R; Albrecht, Brian K; Cochran, Andrea G.
Afiliação
  • Taylor AM; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Bailey C; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Belmont LD; Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States.
  • Campbell R; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Cantone N; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Côté A; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Crawford TD; Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States.
  • Cummings R; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • DeMent K; Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States.
  • Duplessis M; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Flynn M; Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States.
  • Good AC; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Huang HR; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Joshi S; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Leblanc Y; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Murray J; Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States.
  • Nasveschuk CG; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Neiss A; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Poy F; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Romero FA; Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States.
  • Sandy P; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Tang Y; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Tsui V; Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States.
  • Zawadzke L; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Sims RJ; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Audia JE; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Bellon SF; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Magnuson SR; Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States.
  • Albrecht BK; Constellation, a Morphosys Company, 215 First Street, Suite 200, Cambridge, Massachusetts 02142, United States.
  • Cochran AG; Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States.
J Med Chem ; 65(16): 11177-11186, 2022 08 25.
Article em En | MEDLINE | ID: mdl-35930799

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / DNA Helicases Limite: Humans Idioma: En Revista: J Med Chem Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / DNA Helicases Limite: Humans Idioma: En Revista: J Med Chem Ano de publicação: 2022 Tipo de documento: Article