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Design, Synthesis, Kinetic Analysis and Pharmacophore-Directed Discovery of 3-Ethylaniline Hybrid Imino-Thiazolidinone as Potential Inhibitor of Carbonic Anhydrase II: An Emerging Biological Target for Treatment of Cancer.
Ahmed, Atteeque; Aziz, Mubashir; Ejaz, Syeda Abida; Channar, Pervaiz Ali; Saeed, Aamer; Zargar, Seema; Wani, Tanveer A; Hamad, Asad; Abbas, Qamar; Raza, Hussain; Kim, Song Ja.
Afiliação
  • Ahmed A; Department of Chemistry, Quaid-I-Azam University, Islamabad 45320, Pakistan.
  • Aziz M; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, The Islamia University of Bahawalpur, Bahawalpur 63100, Pakistan.
  • Ejaz SA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, The Islamia University of Bahawalpur, Bahawalpur 63100, Pakistan.
  • Channar PA; Department of Basic Sciences and Humanities, Faculty of Information Science and Humanities, Dawood University of Engineering and Technology, Karachi 74800, Pakistan.
  • Saeed A; Department of Chemistry, Quaid-I-Azam University, Islamabad 45320, Pakistan.
  • Zargar S; Department of Biochemistry, College of Science, King Saud University, P.O. Box 22452, Riyadh 11451, Saudi Arabia.
  • Wani TA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
  • Hamad A; Faculty of Pharmacy, Grand Asian University Sialkot, Sialkot 51310, Pakistan.
  • Abbas Q; Department of Biology, College of Science, University of Bahrain, Sakhir 32038, Bahrain.
  • Raza H; College of Natural Sciences, Department of Biological Sciences, Kongju National University, Gongju 32588, Republic of Korea.
  • Kim SJ; College of Natural Sciences, Department of Biological Sciences, Kongju National University, Gongju 32588, Republic of Korea.
Biomolecules ; 12(11)2022 11 16.
Article em En | MEDLINE | ID: mdl-36421710

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Anidrase Carbônica II / Neoplasias Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: Biomolecules Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Anidrase Carbônica II / Neoplasias Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: Biomolecules Ano de publicação: 2022 Tipo de documento: Article