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Tautomer-Specific Deacylation and Ω-Loop Flexibility Explain the Carbapenem-Hydrolyzing Broad-Spectrum Activity of the KPC-2 ß-Lactamase.
Tooke, Catherine L; Hinchliffe, Philip; Beer, Michael; Zinovjev, Kirill; Colenso, Charlotte K; Schofield, Christopher J; Mulholland, Adrian J; Spencer, James.
Afiliação
  • Tooke CL; School of Cellular and Molecular Medicine, Biomedical Sciences Building, University Walk, University of Bristol, Bristol BS8 1TD, United Kingdom.
  • Hinchliffe P; School of Cellular and Molecular Medicine, Biomedical Sciences Building, University Walk, University of Bristol, Bristol BS8 1TD, United Kingdom.
  • Beer M; School of Cellular and Molecular Medicine, Biomedical Sciences Building, University Walk, University of Bristol, Bristol BS8 1TD, United Kingdom.
  • Zinovjev K; Centre for Computational Chemistry, School of Chemistry, Cantock's Close, University of Bristol, Bristol BS8 1TS, United Kingdom.
  • Colenso CK; School of Biochemistry, Biomedical Sciences Building, University Walk, University of Bristol, Bristol BS8 1TD, United Kingdom.
  • Schofield CJ; Departamento de Química Física, Universitat de València, Burjassot 46100, Comunitat Valenciana, Spain.
  • Mulholland AJ; School of Cellular and Molecular Medicine, Biomedical Sciences Building, University Walk, University of Bristol, Bristol BS8 1TD, United Kingdom.
  • Spencer J; Centre for Computational Chemistry, School of Chemistry, Cantock's Close, University of Bristol, Bristol BS8 1TS, United Kingdom.
J Am Chem Soc ; 145(13): 7166-7180, 2023 04 05.
Article em En | MEDLINE | ID: mdl-36972204

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 3_ND Base de dados: MEDLINE Assunto principal: Carbapenêmicos / Antibacterianos Idioma: En Revista: J Am Chem Soc Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Contexto em Saúde: 3_ND Base de dados: MEDLINE Assunto principal: Carbapenêmicos / Antibacterianos Idioma: En Revista: J Am Chem Soc Ano de publicação: 2023 Tipo de documento: Article