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Radiometal Complexes as Pharmacokinetic Modifiers: A Potent 68Ga-Labeled Gastrin-Releasing Peptide Receptor Antagonist Based on the Macrocyclic Metal Chelator NODIA-Me.
Schreck, Moritz-Valentin; Burgard, Caroline; Schmidtke, Alexander; Hierlmeier, Ina; Stemler, Tobias; Maus, Stephan; Rosar, Florian; Jung, Martin; Speicher, Andreas; Ezziddin, Samer; Holland, Jason P; Bartholomä, Mark D.
Afiliação
  • Schreck MV; Department of Nuclear Medicine, Saarland University-Medical Center, Kirrbergerstrasse, D-66421 Homburg, Germany.
  • Burgard C; Department of Nuclear Medicine, Saarland University-Medical Center, Kirrbergerstrasse, D-66421 Homburg, Germany.
  • Schmidtke A; Department of Nuclear Medicine, Saarland University-Medical Center, Kirrbergerstrasse, D-66421 Homburg, Germany.
  • Hierlmeier I; Department of Nuclear Medicine, Saarland University-Medical Center, Kirrbergerstrasse, D-66421 Homburg, Germany.
  • Stemler T; Department of Nuclear Medicine, Saarland University-Medical Center, Kirrbergerstrasse, D-66421 Homburg, Germany.
  • Maus S; Department of Nuclear Medicine, Saarland University-Medical Center, Kirrbergerstrasse, D-66421 Homburg, Germany.
  • Rosar F; Department of Nuclear Medicine, Saarland University-Medical Center, Kirrbergerstrasse, D-66421 Homburg, Germany.
  • Jung M; Department of Medical Biochemistry and Molecular Biology, Saarland University, D-66421 Homburg, Germany.
  • Speicher A; Department of Organic Chemistry, Saarland University, D-66123 Saarbrücken, Germany.
  • Ezziddin S; Department of Nuclear Medicine, Saarland University-Medical Center, Kirrbergerstrasse, D-66421 Homburg, Germany.
  • Holland JP; Department of Chemistry, University of Zurich, Winterthurerstrasse 190, CH-8057 Zurich, Switzerland.
  • Bartholomä MD; Department of Nuclear Medicine, Saarland University-Medical Center, Kirrbergerstrasse, D-66421 Homburg, Germany.
Mol Pharm ; 20(12): 6463-6473, 2023 Dec 04.
Article em En | MEDLINE | ID: mdl-37978936

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Neoplasias da Próstata / Neoplasias da Mama Limite: Animals / Humans / Male Idioma: En Revista: Mol Pharm Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Neoplasias da Próstata / Neoplasias da Mama Limite: Animals / Humans / Male Idioma: En Revista: Mol Pharm Ano de publicação: 2023 Tipo de documento: Article