An HPLC assay for the norditerpenoid alkaloid methyllycaconitine, a potent nicotinic acetylcholine receptor antagonist.
J Pharm Biomed Anal
; 13(12): 1541-44, 1995 Nov.
Article
em En
| MEDLINE
| ID: mdl-8788140
The extremely potent and selective nicotinic acetylcholine receptor antagonist methyllycaconitine, MLA, and related norditerpene alkaloids are finding increasing use as neurochemical probes and as targets for structure-activity relationship studies. In this work, an assay procedure for MLA which utilises ion suppression reverse-phase HPLC with UV absorbance detection at 270 nm is described. The method detected 280 ng MLA on column.
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Coleções:
01-internacional
Base de dados:
MEDLINE
Assunto principal:
Aconitina
/
Antagonistas Nicotínicos
Idioma:
En
Revista:
J Pharm Biomed Anal
Ano de publicação:
1995
Tipo de documento:
Article