Detalhe da pesquisa
1.
Synthesis of metronidazole based thiazolidinone analogs as promising antiamoebic agents.
Bioorg Med Chem Lett
; 30(23): 127549, 2020 12 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-32927029
2.
Effect of triazole-tryptophan hybrid on the conformation stability of bovine serum albumin.
Luminescence
; 33(3): 464-474, 2018 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-29314579
3.
New antiprotozoal agents: Synthesis and biological evaluation of different 4-(7-chloroquinolin-4-yl) piperazin-1-yl)pyrrolidin-2-yl)methanone derivatives.
Bioorg Med Chem Lett
; 27(3): 460-465, 2017 02 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28027871
4.
Anti-leishmanial and cytotoxic activities of amino acid-triazole hybrids: Synthesis, biological evaluation, molecular docking and in silico physico-chemical properties.
Bioorg Med Chem Lett
; 27(9): 1886-1891, 2017 05 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28359789
5.
Recent progress on the discovery of antiamoebic agents.
Bioorg Med Chem Lett
; 26(21): 5149-5159, 2016 11 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-27707603
6.
Effect of novel triazole-amino acid hybrids on growth and virulence of Candida species: in vitro and in vivo studies.
Org Biomol Chem
; 14(45): 10599-10619, 2016 Dec 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-27735963
7.
Monocyclic ß-lactam and unexpected oxazinone formation: synthesis, crystal structure, docking studies and antibacterial evaluation.
J Enzyme Inhib Med Chem
; 31(5): 834-52, 2016 Oct.
Artigo
em Inglês
| MEDLINE | ID: mdl-26133357
8.
Metronidazole hydrazone conjugates: Design, synthesis, antiamoebic and molecular docking studies.
Bioorg Med Chem Lett
; 25(17): 3545-9, 2015 Sep 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-26174554
9.
Synthesis and evaluation of 7-chloro-4-(piperazin-1-yl)quinoline-sulfonamide as hybrid antiprotozoal agents.
Bioorg Med Chem
; 21(11): 3080-9, 2013 Jun 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-23602620
10.
Discovery of Novel Hydroxyimine-Tethered Benzenesulfonamides as Potential Human Carbonic Anhydrase IX/XII Inhibitors.
ACS Med Chem Lett
; 14(6): 810-819, 2023 Jun 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-37312840
11.
Metronidazole thiosalicylate conjugates: synthesis, crystal structure, docking studies and antiamoebic activity.
Bioorg Med Chem Lett
; 22(17): 5694-9, 2012 Sep 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-22832309
12.
Thiosemicarbazone fragment embedded within 1,2,4-triazole ring as inhibitors of Entamoeba histolytica.
Bioorg Med Chem Lett
; 22(8): 2768-71, 2012 Apr 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22444681
13.
Synthesis and Anticancer Evaluation of Novel Indole Based Arylsulfonylhydrazides against Human Breast Cancer Cells.
ACS Omega
; 7(46): 42036-42043, 2022 Nov 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-36440122
14.
Synthesis, characterization, antiamoebic activity and cytotoxicity of new pyrazolo[3, 4-d]pyrimidine-6-one derivatives.
J Enzyme Inhib Med Chem
; 26(4): 472-9, 2011 Aug.
Artigo
em Inglês
| MEDLINE | ID: mdl-21054147
15.
Advances in Drug Discovery against Neglected Tropical Diseases: Human African and American Trypanosomiasis.
Curr Med Chem
; 28(36): 7544-7582, 2021.
Artigo
em Inglês
| MEDLINE | ID: mdl-33949927
16.
Deciphering the key heterocyclic scaffolds in targeting microtubules, kinases and carbonic anhydrases for cancer drug development.
Pharmacol Ther
; 225: 107860, 2021 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-33895188
17.
Development of Oxadiazole-Sulfonamide-Based Compounds as Potential Antibacterial Agents.
ACS Omega
; 6(42): 27798-27813, 2021 Oct 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-34722980
18.
Structure-activity relationships of mononuclear metal-thiosemicarbazone complexes endowed with potent antiplasmodial and antiamoebic activities.
Bioorg Med Chem
; 18(18): 6857-64, 2010 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20719524
19.
Design and Development of Small-Molecule Arylaldoxime/5-Nitroimidazole Hybrids as Potent Inhibitors of MARK4: A Promising Approach for Target-Based Cancer Therapy.
ACS Omega
; 5(36): 22759-22771, 2020 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-32954123
20.
Discovery of 4-(2-(dimethylamino)ethoxy)benzohydrazide derivatives as prospective microtubule affinity regulating kinase 4 inhibitors.
RSC Adv
; 10(34): 20129-20137, 2020 May 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-35520423