Detalhe da pesquisa
1.
Radiofluorination of oxazole-carboxamides for preclinical PET neuroimaging of GSK-3.
J Fluor Chem
; 2452021 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-33840834
2.
Efficient radiosynthesis and preclinical evaluation of [18 F]FOMPyD as a positron emission tomography tracer candidate for TrkB/C receptor imaging.
J Labelled Comp Radiopharm
; 63(3): 144-150, 2020 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-31919878
3.
Synthesis and preclinical evaluation of [18F]FSL25.1188, a reversible PET radioligand for monoamine oxidase-B.
Bioorg Med Chem Lett
; 29(13): 1624-1627, 2019 07 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-31060887
4.
Emerging PET Radiotracers and Targets for Imaging of Neuroinflammation in Neurodegenerative Diseases: Outlook Beyond TSPO.
Mol Imaging
; 17: 1536012118792317, 2018.
Artigo
em Inglês
| MEDLINE | ID: mdl-30203712
5.
Metal Protein-Attenuating Compound for PET Neuroimaging: Synthesis and Preclinical Evaluation of [11C]PBT2.
Mol Pharm
; 15(2): 695-702, 2018 02 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-29298483
6.
Automated synthesis of PET radiotracers by copper-mediated 18 F-fluorination of organoborons: Importance of the order of addition and competing protodeborylation.
J Labelled Comp Radiopharm
; 61(3): 228-236, 2018 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-29143408
7.
Design and synthesis of a fluorinated quinazoline-based type-II Trk inhibitor as a scaffold for PET radiotracer development.
Bioorg Med Chem Lett
; 27(12): 2771-2775, 2017 06 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-28476569
8.
Discovery of PET radiopharmaceuticals at the academia-industry interface.
Drug Discov Today Technol
; 25: 19-26, 2017 Nov.
Artigo
em Inglês
| MEDLINE | ID: mdl-29233263
9.
From Unorthodox to Established: The Current Status of (18)F-Trifluoroborate- and (18)F-SiFA-Based Radiopharmaceuticals in PET Nuclear Imaging.
Bioconjug Chem
; 27(2): 267-79, 2016 Feb 17.
Artigo
em Inglês
| MEDLINE | ID: mdl-26566577
10.
Recent Advances in the Development and Application of Radiolabeled Kinase Inhibitors for PET Imaging.
Molecules
; 20(12): 22000-27, 2015 Dec 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-26690113
11.
5-(4-((4-[(18)F]Fluorobenzyl)oxy)-3-methoxybenzyl)pyrimidine-2,4-diamine: a selective dual inhibitor for potential PET imaging of Trk/CSF-1R.
Bioorg Med Chem Lett
; 24(20): 4784-90, 2014 Oct 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-25257201
12.
Direct one-step labeling of cysteine residues on peptides with [(11)C]methyl triflate for the synthesis of PET radiopharmaceuticals.
Amino Acids
; 45(5): 1097-108, 2013 Nov.
Artigo
em Inglês
| MEDLINE | ID: mdl-23921782
13.
Towards tropomyosin-related kinase B (TrkB) receptor ligands for brain imaging with PET: radiosynthesis and evaluation of 2-(4-[(18)F]fluorophenyl)-7,8-dihydroxy-4H-chromen-4-one and 2-(4-([N-methyl-(11)C]-dimethylamino)phenyl)-7,8-dihydroxy-4H-chromen-4-one.
Bioorg Med Chem
; 21(24): 7816-29, 2013 Dec 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-24183588
14.
Preliminary Evaluations of [11C]Verubulin: Implications for Microtubule Imaging With PET.
Front Neurosci
; 15: 725873, 2021.
Artigo
em Inglês
| MEDLINE | ID: mdl-34566568
15.
Probing Anti-inflammatory Properties Independent of NF-κB Through Conformational Constraint of Peptide-Based Interleukin-1 Receptor Biased Ligands.
Front Chem
; 7: 23, 2019.
Artigo
em Inglês
| MEDLINE | ID: mdl-30815434
16.
First-in-Human Brain Imaging of [18F]TRACK, a PET tracer for Tropomyosin Receptor Kinases.
ACS Chem Neurosci
; 10(6): 2697-2702, 2019 06 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-31017386
17.
Radioligands for Tropomyosin Receptor Kinase (Trk) Positron Emission Tomography Imaging.
Pharmaceuticals (Basel)
; 12(1)2019 Jan 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-30609832
18.
Structural Basis for Achieving GSK-3ß Inhibition with High Potency, Selectivity, and Brain Exposure for Positron Emission Tomography Imaging and Drug Discovery.
J Med Chem
; 62(21): 9600-9617, 2019 11 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-31535859
19.
Fluorine-18: an untapped resource in inorganic chemistry.
Chem Commun (Camb)
; 54(84): 11835-11842, 2018 Oct 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-30191929
20.
Recent Advances in 18F Radiochemistry: A Focus on B-18F, Si-18F, Al-18F, and C-18F Radiofluorination via Spirocyclic Iodonium Ylides.
J Nucl Med
; 59(4): 568-572, 2018 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-29284673