Detalhe da pesquisa
1.
Discovery of Proline-Based p300/CBP Inhibitors Using DNA-Encoded Library Technology in Combination with High-Throughput Screening.
J Med Chem
; 65(21): 14391-14408, 2022 11 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-36302181
2.
Cell-Based Drug Discovery: Identification and Optimization of Small Molecules that Reduce c-MYC Protein Levels in Cells.
J Med Chem
; 64(21): 16056-16087, 2021 11 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-34669409
3.
Identification of 5α, 6α-epoxycholesterol as a novel modulator of liver X receptor activity.
Mol Pharmacol
; 78(6): 1046-58, 2010 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-20837678
4.
1-Methyl-1H-pyrrole-2-carbonitrile containing tetrahydronaphthalene derivatives as non-steroidal progesterone receptor antagonists.
Bioorg Med Chem Lett
; 20(16): 4816-8, 2010 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20638844
5.
Differential biochemical and cellular actions of Premarin estrogens: distinct pharmacology of bazedoxifene-conjugated estrogens combination.
Mol Endocrinol
; 23(1): 74-85, 2009 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-19036900
6.
LXR ligand lowers LDL cholesterol in primates, is lipid neutral in hamster, and reduces atherosclerosis in mouse.
J Lipid Res
; 50(12): 2358-70, 2009 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-19318684
7.
5-Aryl indanones and derivatives as non-steroidal progesterone receptor modulators.
Bioorg Med Chem Lett
; 19(23): 6666-9, 2009 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-19864132
8.
Characterization of ligands for thyroid receptor subtypes and their interactions with co-regulators.
Steroids
; 74(2): 270-6, 2009 Feb.
Artigo
em Inglês
| MEDLINE | ID: mdl-19073200
9.
The lecanindoles, nonsteroidal progestins from the terrestrial fungus Verticillium lecanii 6144.
J Nat Prod
; 72(11): 1944-8, 2009 Nov.
Artigo
em Inglês
| MEDLINE | ID: mdl-19863083
10.
1,5-Dihydro-benzo[e][1,4]oxazepin-2(1H)-ones containing a 7-(5'-cyanopyrrol-2-yl) group as nonsteroidal progesterone receptor modulators.
Bioorg Med Chem Lett
; 18(18): 5015-7, 2008 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-18722119
11.
7-aryl 1,5-dihydro-benzo[e][1,4]oxazepin-2-ones and analogs as non-steroidal progesterone receptor antagonists.
Bioorg Med Chem
; 16(13): 6589-600, 2008 Jul 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-18504132
12.
Identification of novel estrogen receptor alpha antagonists.
J Steroid Biochem Mol Biol
; 88(4-5): 351-60, 2004 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-15145444
13.
Discovery of a novel mechanism of steroid receptor antagonism: WAY-255348 modulates progesterone receptor cellular localization and promoter interactions.
Biochem Pharmacol
; 82(11): 1709-19, 2011 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21854761
14.
Identification of phenylsulfone-substituted quinoxaline (WYE-672) as a tissue selective liver X-receptor (LXR) agonist.
J Med Chem
; 53(8): 3296-304, 2010 Apr 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-20350005
15.
Novel progesterone receptor modulators with gene selective and context-dependent partial agonism.
Biochem Pharmacol
; 77(2): 204-15, 2009 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-19013437