Detalhe da pesquisa
1.
SAR towards indoline and 3-azaindoline classes of IDO1 inhibitors.
Bioorg Med Chem Lett
; 47: 128214, 2021 09 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-34166782
2.
Structural characterization of nonactive site, TrkA-selective kinase inhibitors.
Proc Natl Acad Sci U S A
; 114(3): E297-E306, 2017 01 17.
Artigo
em Inglês
| MEDLINE | ID: mdl-28039433
3.
Carbamate and N-Pyrimidine Mitigate Amide Hydrolysis: Structure-Based Drug Design of Tetrahydroquinoline IDO1 Inhibitors.
ACS Med Chem Lett
; 12(3): 389-396, 2021 Mar 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-33738066
4.
Targeting RNA with Small Molecules: Identification of Selective, RNA-Binding Small Molecules Occupying Drug-Like Chemical Space.
SLAS Discov
; 25(4): 384-396, 2020 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-31701793
5.
Identification of G-Quadruplex-Binding Inhibitors of Myc Expression through Affinity Selection-Mass Spectrometry.
SLAS Discov
; 24(2): 142-157, 2019 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-30204533
6.
Discovery of Selective RNA-Binding Small Molecules by Affinity-Selection Mass Spectrometry.
ACS Chem Biol
; 13(3): 820-831, 2018 03 16.
Artigo
em Inglês
| MEDLINE | ID: mdl-29412640
7.
Linking High-Throughput Screens to Identify MoAs and Novel Inhibitors of Mycobacterium tuberculosis Dihydrofolate Reductase.
ACS Chem Biol
; 12(9): 2448-2456, 2017 09 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-28806050
8.
Integration of Affinity Selection-Mass Spectrometry and Functional Cell-Based Assays to Rapidly Triage Druggable Target Space within the NF-κB Pathway.
J Biomol Screen
; 21(6): 608-19, 2016 Jul.
Artigo
em Inglês
| MEDLINE | ID: mdl-26969322