Detalhe da pesquisa
1.
Small-molecule modulators of PXR and CAR.
Biochim Biophys Acta
; 1859(9): 1141-1154, 2016 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-26921498
2.
Identification and Characterization of CINPA1 Metabolites Facilitates Structure-Activity Studies of the Constitutive Androstane Receptor.
Drug Metab Dispos
; 44(11): 1759-1770, 2016 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-27519550
3.
CINPA1 is an inhibitor of constitutive androstane receptor that does not activate pregnane X receptor.
Mol Pharmacol
; 87(5): 878-89, 2015 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-25762023
4.
A competitive inhibitor that reduces recruitment of androgen receptor to androgen-responsive genes.
J Biol Chem
; 287(28): 23368-80, 2012 Jul 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-22589544
5.
Small molecule inhibitors as probes for estrogen and androgen receptor action.
J Biol Chem
; 286(6): 4043-8, 2011 Feb 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-21149443
6.
A noncompetitive small molecule inhibitor of estrogen-regulated gene expression and breast cancer cell growth that enhances proteasome-dependent degradation of estrogen receptor {alpha}.
J Biol Chem
; 285(53): 41863-73, 2010 Dec 31.
Artigo
em Inglês
| MEDLINE | ID: mdl-21041310
7.
CINPA1 binds directly to constitutive androstane receptor and inhibits its activity.
Biochem Pharmacol
; 152: 211-223, 2018 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-29608908
8.
The orphan nuclear receptor NR4A2 is part of a p53-microRNA-34 network.
Sci Rep
; 6: 25108, 2016 04 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-27121375
9.
Small-molecule modulators of the constitutive androstane receptor.
Expert Opin Drug Metab Toxicol
; 11(7): 1099-114, 2015 Jul.
Artigo
em Inglês
| MEDLINE | ID: mdl-25979168
10.
A new small molecule inhibitor of estrogen receptor alpha binding to estrogen response elements blocks estrogen-dependent growth of cancer cells.
J Biol Chem
; 283(19): 12819-30, 2008 May 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-18337247