Detalhe da pesquisa
1.
Imaging EGFR and HER2 by PET and SPECT: a review.
Med Res Rev
; 34(3): 596-643, 2014 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-24037872
2.
4,4'-Unsymmetrically substituted 3,3'-biphenyl alpha helical proteomimetics as potential coactivator binding inhibitors.
Bioorg Med Chem
; 22(2): 917-26, 2014 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-24360824
3.
Synthesis and preliminary evaluation steroidal antiestrogen-geldanamycin conjugates.
Bioorg Med Chem Lett
; 23(12): 3635-9, 2013 Jun 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-23648180
4.
Targeting the estrogen receptor using steroid-therapeutic drug conjugates (hybrids).
Bioconjug Chem
; 23(11): 2139-58, 2012 Nov 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-23036054
5.
Design, synthesis, and initial biological evaluation of a steroidal anti-estrogen-doxorubicin bioconjugate for targeting estrogen receptor-positive breast cancer cells.
Bioconjug Chem
; 23(4): 785-95, 2012 Apr 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-22404783
6.
3,3'-Disubstituted bipolar biphenyls as inhibitors of nuclear receptor coactivator binding.
Bioorg Med Chem Lett
; 22(21): 6587-90, 2012 Nov 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-23017882
7.
Synthesis of a spin-labeled anti-estrogen as a dynamic motion probe for the estrogen receptor ligand binding domain.
Bioorg Med Chem Lett
; 22(4): 1743-6, 2012 Feb 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22257894
8.
Synthesis and evaluation of 4-(substituted styryl/alkenyl)-3,5-bis(4-hydroxyphenyl)-isoxazoles as ligands for the estrogen receptor.
Bioorg Med Chem Lett
; 22(18): 5999-6003, 2012 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22906893
9.
Targeting the estrogen receptor with metal-carbonyl derivatives of estradiol.
Bioorg Med Chem Lett
; 22(4): 1670-3, 2012 Feb 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22277281
10.
Synthesis and evaluation of 17α-E-20-(heteroaryl)norpregn-1,3,5(10),20 tetraene-3,17ß-diols [17α-(heteroaryl)vinyl estradiols] as ligands for the estrogen receptor-α ligand binding domain (ERα-LBD).
Bioorg Med Chem Lett
; 22(2): 977-9, 2012 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22178552
11.
Convergent synthesis of a steroidal antiestrogen-mitomycin C hybrid using "click" chemistry.
Org Biomol Chem
; 10(42): 8501-8, 2012 Nov 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-23007562
12.
Synthesis and evaluation of 11ß-(4-substituted phenyl) estradiol analogs: transition from estrogen receptor agonists to antagonists.
Bioorg Med Chem
; 20(12): 3768-80, 2012 Jun 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22608920
13.
Review of fluorescent steroidal ligands for the estrogen receptor 1995-2018.
Steroids
; 144: 30-46, 2019 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-30738074
14.
Design and synthesis of fluorescently labeled steroidal antiestrogens.
Steroids
; 145: 39-46, 2019 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-30797876
15.
Synthesis of benzoylbenzamide derivatives of 17α-E-vinyl estradiol and evaluation as ligands for the estrogen receptor-α ligand binding domain.
Steroids
; 144: 15-20, 2019 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-30738075
16.
Synthesis and evaluation of isomeric (17alpha,20E)-11beta-methoxy-21-(trifluoromethylphenyl)-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diols as ERalpha-hormone binding domain ligands: effect of the methoxy group on receptor binding and uterotrophic growth.
J Med Chem
; 50(3): 472-9, 2007 Feb 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-17266199
17.
Synthesis and evaluation of (17alpha,20Z)-21-(4-substituted-phenyl)-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diols as ligands for the estrogen receptor-alpha hormone binding domain: comparison with 20E-isomers.
J Med Chem
; 48(13): 4300-11, 2005 Jun 30.
Artigo
em Inglês
| MEDLINE | ID: mdl-15974584
18.
Synthesis and evaluation of 2-halogenated-1,1-bis(4-hydroxyphenyl)-2-(3-hydroxyphenyl)-ethylenes as potential estrogen receptor-targeted radiodiagnostic and radiotherapeutic agents.
Steroids
; 96: 50-62, 2015 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-25637676
19.
Synthesis and evaluation of 17alpha-20E-21-(4-substituted phenyl)-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diols as probes for the estrogen receptor alpha hormone binding domain.
J Med Chem
; 46(14): 2865-76, 2003 Jul 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-12825929
20.
Evaluation of 17alpha-E-(trifluoromethylphenyl)vinyl estradiols as novel estrogen receptor ligands.
Steroids
; 68(2): 143-8, 2003 Feb.
Artigo
em Inglês
| MEDLINE | ID: mdl-12606005