Detalhe da pesquisa
1.
Unsymmetrical Bisquinolines with High Potency against P. falciparum Malaria.
Molecules
; 25(9)2020 May 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-32397659
2.
ELQ-331 as a prototype for extremely durable chemoprotection against malaria.
Malar J
; 18(1): 291, 2019 Aug 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-31455339
3.
Simplified Reversed Chloroquines To Overcome Malaria Resistance to Quinoline-Based Drugs.
Antimicrob Agents Chemother
; 61(5)2017 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-28193646
4.
Atovaquone and ELQ-300 Combination Therapy as a Novel Dual-Site Cytochrome bc1 Inhibition Strategy for Malaria.
Antimicrob Agents Chemother
; 60(8): 4853-9, 2016 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-27270285
5.
Interrogating the Tailoring Steps of Pactamycin Biosynthesis and Accessing New Pactamycin Analogues.
Chembiochem
; 17(17): 1585-8, 2016 09 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-27305101
6.
ELQ-300 prodrugs for enhanced delivery and single-dose cure of malaria.
Antimicrob Agents Chemother
; 59(9): 5555-60, 2015 Sep.
Artigo
em Inglês
| MEDLINE | ID: mdl-26124159
7.
Depsipeptide companeramides from a Panamanian marine cyanobacterium associated with the coibamide producer.
J Nat Prod
; 78(3): 413-20, 2015 Mar 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-25562664
8.
Discovery of dual function acridones as a new antimalarial chemotype.
Nature
; 459(7244): 270-3, 2009 May 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-19357645
9.
Discovery and Optimization of Tambjamines as a Novel Class of Antileishmanial Agents.
J Med Chem
; 67(10): 8323-8345, 2024 May 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-38722757
10.
Optimization of endochin-like quinolones for antimalarial activity.
Exp Parasitol
; 127(2): 545-51, 2011 Feb.
Artigo
em Inglês
| MEDLINE | ID: mdl-21040724
11.
Total Synthesis and Antimalarial Activity of 2-(p-Hydroxybenzyl)-prodigiosins, Isoheptylprodigiosin, and Geometric Isomers of Tambjamine MYP1 Isolated from Marine Bacteria.
J Med Chem
; 64(12): 8739-8754, 2021 06 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-34111350
12.
Acridones Are Highly Potent Inhibitors of Toxoplasma gondii Tachyzoites.
ACS Infect Dis
; 7(7): 1877-1884, 2021 07 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-33723998
13.
Lead Optimization of Second-Generation Acridones as Broad-Spectrum Antimalarials.
J Med Chem
; 63(11): 6179-6202, 2020 06 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-32390431
14.
Boron Trifluoride Etherate Promoted Microwave-Assisted Synthesis of Antimalarial Acridones.
RSC Adv
; 9(72): 42284-42293, 2019.
Artigo
em Inglês
| MEDLINE | ID: mdl-35321096
15.
Discovery and Structural Optimization of Acridones as Broad-Spectrum Antimalarials.
J Med Chem
; 62(7): 3475-3502, 2019 04 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-30852885
16.
Synthesis and heme-binding correlation with antimalarial activity of 3,6-bis-(omega-N,N-diethylaminoamyloxy)-4,5-difluoroxanthone.
Bioorg Med Chem
; 16(3): 1174-83, 2008 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-18023189
17.
Alkoxycarbonate Ester Prodrugs of Preclinical Drug Candidate ELQ-300 for Prophylaxis and Treatment of Malaria.
ACS Infect Dis
; 3(10): 728-735, 2017 10 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-28927276
18.
Diphenylether-Modified 1,2-Diamines with Improved Drug Properties for Development against Mycobacterium tuberculosis.
ACS Infect Dis
; 2(7): 500-8, 2016 07 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-27626102
19.
Inhibition of cytochrome bc1 as a strategy for single-dose, multi-stage antimalarial therapy.
Am J Trop Med Hyg
; 92(6): 1195-201, 2015 Jun.
Artigo
em Inglês
| MEDLINE | ID: mdl-25918204
20.
Mutasynthesis of fluorinated pactamycin analogues and their antimalarial activity.
Org Lett
; 15(7): 1678-81, 2013 Apr 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-23521145