Detalhe da pesquisa
1.
Selective Activation of D3 Dopamine Receptors Ameliorates DOI-Induced Head Twitching Accompanied by Changes in Corticostriatal Processing.
Int J Mol Sci
; 24(11)2023 May 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-37298250
2.
Design and Synthesis of D3R Bitopic Ligands with Flexible Secondary Binding Fragments: Radioligand Binding and Computational Chemistry Studies.
Molecules
; 29(1)2023 Dec 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-38202706
3.
Design and Synthesis of Conformationally Flexible Scaffold as Bitopic Ligands for Potent D3-Selective Antagonists.
Int J Mol Sci
; 24(1)2022 Dec 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-36613875
4.
Factors Governing Selectivity of Dopamine Receptor Binding Compounds for D2R and D3R Subtypes.
J Chem Inf Model
; 61(6): 2829-2843, 2021 06 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-33988991
5.
Evaluation of Substituted N-Phenylpiperazine Analogs as D3 vs. D2 Dopamine Receptor Subtype Selective Ligands.
Molecules
; 26(11)2021 May 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-34073405
6.
Design, synthesis, and evaluation of N-(4-(4-phenyl piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamides as selective dopamine D3 receptor ligands.
Bioorg Med Chem Lett
; 29(18): 2690-2694, 2019 09 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-31387791
7.
Challenges in the development of dopamine D2- and D3-selective radiotracers for PET imaging studies.
J Labelled Comp Radiopharm
; 61(3): 291-298, 2018 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-28857231
8.
Synthesis, pharmacological evaluation and molecular modeling studies of triazole containing dopamine D3 receptor ligands.
Bioorg Med Chem Lett
; 25(3): 519-23, 2015 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-25556097
9.
Characterization of [(3) H]LS-3-134, a novel arylamide phenylpiperazine D3 dopamine receptor selective radioligand.
J Neurochem
; 131(4): 418-31, 2014 Nov.
Artigo
em Inglês
| MEDLINE | ID: mdl-25041389
10.
In vitro characterization of [125I]HY-3-24, a selective ligand for the dopamine D3 receptor.
Front Neurosci
; 18: 1380009, 2024.
Artigo
em Inglês
| MEDLINE | ID: mdl-38655111
11.
Reduction of cocaine self-administration and D3 receptor-mediated behavior by two novel dopamine D3 receptor-selective partial agonists, OS-3-106 and WW-III-55.
J Pharmacol Exp Ther
; 347(2): 410-23, 2013 Nov.
Artigo
em Inglês
| MEDLINE | ID: mdl-24018640
12.
Fos expression in response to dopamine D3-preferring phenylpiperazine drugs given with and without cocaine.
Synapse
; 67(12): 847-55, 2013 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-23766142
13.
Evaluation of N-phenyl homopiperazine analogs as potential dopamine D3 receptor selective ligands.
Bioorg Med Chem
; 21(11): 2988-98, 2013 Jun 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-23618707
14.
The effect of SV 293, a D2 dopamine receptor-selective antagonist, on D2 receptor-mediated GIRK channel activation and adenylyl cyclase inhibition.
Pharmacology
; 92(1-2): 84-9, 2013.
Artigo
em Inglês
| MEDLINE | ID: mdl-23942137
15.
Synthesis of bitopic ligands based on fallypride and evaluation of their affinity and selectivity towards dopamine D2 and D3 receptors.
Eur J Med Chem
; 261: 115751, 2023 Dec 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-37688938
16.
Synthesis and Pharmacological Characterization of a Difluorinated Analogue of Reduced Haloperidol as a Sigma-1 Receptor Ligand.
ACS Chem Neurosci
; 14(5): 947-957, 2023 03 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-36780706
17.
Decreased striatal dopamine receptor binding in primary focal dystonia: a D2 or D3 defect?
Mov Disord
; 26(1): 100-6, 2011 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-20960437
18.
Endogenous dopamine (DA) competes with the binding of a radiolabeled D3 receptor partial agonist in vivo: a positron emission tomography study.
Synapse
; 65(8): 724-32, 2011 Aug.
Artigo
em Inglês
| MEDLINE | ID: mdl-21132811
19.
Synthesis and characterization of selective dopamine D2 receptor ligands using aripiprazole as the lead compound.
Bioorg Med Chem
; 19(11): 3502-11, 2011 Jun 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21536445
20.
Interaction of Ligands for PET with the Dopamine D3 Receptor: In Silico and In Vitro Methods.
Biomolecules
; 11(4)2021 04 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-33918451