Detalhe da pesquisa
1.
Turning the Imidazole Core into Three-Dimensional Ring Systems: Mild Organocatalytic Entry to Enantiopure 6,7-Dihydrobenzimidazoles.
Chemistry
; 29(43): e202301200, 2023 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-37204016
2.
Nintedanib-αVß6 Integrin Ligand Conjugates Reduce TGFß-Induced EMT in Human Non-Small Cell Lung Cancer.
Int J Mol Sci
; 24(2)2023 Jan 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-36674990
3.
Novel Polymyxin-Inspired Peptidomimetics Targeting the SARS-CoV-2 Spike:hACE2 Interface.
Int J Mol Sci
; 24(10)2023 May 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-37240111
4.
New Developments of the Principle of Vinylogy as Applied to π-Extended Enolate-Type Donor Systems.
Chem Rev
; 120(5): 2448-2612, 2020 03 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-32040305
5.
New 4-Aminoproline-Based Small Molecule Cyclopeptidomimetics as Potential Modulators of α4ß1 Integrin.
Molecules
; 26(19)2021 Oct 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-34641610
6.
Shifting Towards αV ß6 Integrin Ligands Using Novel Aminoproline-Based Cyclic Peptidomimetics.
Chemistry
; 26(59): 13468-13475, 2020 Oct 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-32634263
7.
Unlocking Access to Enantiopure Fused Uracils by Chemodivergent [4+2] Cross-Cycloadditions: DFT-Supported Homo-Synergistic Organocatalytic Approach.
Angew Chem Int Ed Engl
; 59(45): 20055-20064, 2020 11 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-32678935
8.
Integrin-targeted AmpRGD sunitinib liposomes as integrated antiangiogenic tools.
Nanomedicine
; 18: 135-145, 2019 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-30849548
9.
Acetaldehyde Silyl Enol Ethers in Enantioselective Mukaiyama Aldol Reactions: Enzyme-Like Organocatalysis in Action.
Angew Chem Int Ed Engl
; 58(11): 3264-3266, 2019 03 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-30730598
10.
Gold Nanoparticles Functionalized with RGD-Semipeptides: A Simple yet Highly Effective Targeting System for αV ß3 Integrins.
Chemistry
; 24(46): 12093-12100, 2018 Aug 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-29923243
11.
Exploiting the Distal Reactivity of Indolyl Methylenemalononitriles: An Asymmetric Organocatalyzed [4+2] Cycloaddition with Enals Enables the Assembly of Elusive Dihydrocarbazoles.
Chemistry
; 22(36): 12637-40, 2016 Aug 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-27348410
12.
Pushing the boundaries of vinylogous reactivity: catalytic enantioselective mukaiyama aldol reactions of highly unsaturated 2-silyloxyindoles.
Chemistry
; 21(17): 6433-42, 2015 Apr 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-25735832
13.
Organocatalytic, Asymmetric Eliminative [4+2] Cycloaddition of Allylidene Malononitriles with Enals: Rapid Entry to Cyclohexadiene-Embedding Linear and Angular Polycycles.
Angew Chem Int Ed Engl
; 54(25): 7386-90, 2015 Jun 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-25950770
14.
Exploring the vinylogous reactivity of cyclohexenylidene malononitriles: switchable regioselectivity in the organocatalytic asymmetric addition to enals giving highly enantioenriched carbabicyclic structures.
J Am Chem Soc
; 136(31): 11107-14, 2014 Aug 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-25032901
15.
Enhancement of the uptake and cytotoxic activity of doxorubicin in cancer cells by novel cRGD-semipeptide-anchoring liposomes.
Mol Pharm
; 11(7): 2280-93, 2014 Jul 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-24819754
16.
Synthesis, structure and inhibitory activity of a stereoisomer of oseltamivir carboxylate.
Org Biomol Chem
; 12(10): 1561-9, 2014 Mar 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-24425043
17.
Design, synthesis, and biological evaluation of novel cRGD-paclitaxel conjugates for integrin-assisted drug delivery.
Bioconjug Chem
; 23(8): 1610-22, 2012 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22770429
18.
Nintedanib-Containing Dual Conjugates Targeting αVß6 Integrin and Tyrosine Kinase Receptors as Potential Antifibrotic Agents.
ACS Omega
; 7(21): 17658-17669, 2022 May 31.
Artigo
em Inglês
| MEDLINE | ID: mdl-35664627
19.
anti-Selective, catalytic asymmetric vinylogous Mukaiyama Mannich reactions of pyrrole-based silyl dienolates with N-aryl aldimines.
J Org Chem
; 76(7): 2248-52, 2011 Apr 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21381711
20.
Diastereo- and enantioselective catalytic vinylogous Mukaiyama-Mannich reactions of pyrrole-based silyl dienolates with alkyl-substituted aldehydes.
J Org Chem
; 76(24): 10291-8, 2011 Dec 16.
Artigo
em Inglês
| MEDLINE | ID: mdl-22059699