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Synthesis and Characterization in Vitro and in Vivo of (l)-(Trimethylsilyl)alanine Containing Neurotensin Analogues.
Fanelli, Roberto; Besserer-Offroy, Élie; René, Adeline; Côté, Jérôme; Tétreault, Pascal; Collerette-Tremblay, Jasmin; Longpré, Jean-Michel; Leduc, Richard; Martinez, Jean; Sarret, Philippe; Cavelier, Florine.
Afiliação
  • Fanelli R; Institut des Biomolécules Max Mousseron, IBMM, UMR-5247, CNRS, Université Montpellier, ENSCM, Place Eugène Bataillon, 34095 Montpellier Cedex 5, France.
  • Besserer-Offroy É; Department of Pharmacology and Physiology, Institut de Pharmacologie de Sherbrooke, Faculty of Medicine and Health Sciences, Université de Sherbrooke , Sherbrooke, Québec J1K 2R1, Canada.
  • René A; Institut des Biomolécules Max Mousseron, IBMM, UMR-5247, CNRS, Université Montpellier, ENSCM, Place Eugène Bataillon, 34095 Montpellier Cedex 5, France.
  • Côté J; Department of Pharmacology and Physiology, Institut de Pharmacologie de Sherbrooke, Faculty of Medicine and Health Sciences, Université de Sherbrooke , Sherbrooke, Québec J1K 2R1, Canada.
  • Tétreault P; Department of Pharmacology and Physiology, Institut de Pharmacologie de Sherbrooke, Faculty of Medicine and Health Sciences, Université de Sherbrooke , Sherbrooke, Québec J1K 2R1, Canada.
  • Collerette-Tremblay J; Department of Pharmacology and Physiology, Institut de Pharmacologie de Sherbrooke, Faculty of Medicine and Health Sciences, Université de Sherbrooke , Sherbrooke, Québec J1K 2R1, Canada.
  • Longpré JM; Department of Pharmacology and Physiology, Institut de Pharmacologie de Sherbrooke, Faculty of Medicine and Health Sciences, Université de Sherbrooke , Sherbrooke, Québec J1K 2R1, Canada.
  • Leduc R; Department of Pharmacology and Physiology, Institut de Pharmacologie de Sherbrooke, Faculty of Medicine and Health Sciences, Université de Sherbrooke , Sherbrooke, Québec J1K 2R1, Canada.
  • Martinez J; Institut des Biomolécules Max Mousseron, IBMM, UMR-5247, CNRS, Université Montpellier, ENSCM, Place Eugène Bataillon, 34095 Montpellier Cedex 5, France.
  • Sarret P; Department of Pharmacology and Physiology, Institut de Pharmacologie de Sherbrooke, Faculty of Medicine and Health Sciences, Université de Sherbrooke , Sherbrooke, Québec J1K 2R1, Canada.
  • Cavelier F; Institut des Biomolécules Max Mousseron, IBMM, UMR-5247, CNRS, Université Montpellier, ENSCM, Place Eugène Bataillon, 34095 Montpellier Cedex 5, France.
J Med Chem ; 58(19): 7785-95, 2015 Oct 08.
Article em En | MEDLINE | ID: mdl-26348111

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Neurotensina / Avaliação Pré-Clínica de Medicamentos Tipo de estudo: Prognostic_studies Limite: Animals Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2015 Tipo de documento: Article País de afiliação: França

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Neurotensina / Avaliação Pré-Clínica de Medicamentos Tipo de estudo: Prognostic_studies Limite: Animals Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2015 Tipo de documento: Article País de afiliação: França