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A cellular chemical probe targeting the chromodomains of Polycomb repressive complex 1.
Stuckey, Jacob I; Dickson, Bradley M; Cheng, Nancy; Liu, Yanli; Norris, Jacqueline L; Cholensky, Stephanie H; Tempel, Wolfram; Qin, Su; Huber, Katherine G; Sagum, Cari; Black, Karynne; Li, Fengling; Huang, Xi-Ping; Roth, Bryan L; Baughman, Brandi M; Senisterra, Guillermo; Pattenden, Samantha G; Vedadi, Masoud; Brown, Peter J; Bedford, Mark T; Min, Jinrong; Arrowsmith, Cheryl H; James, Lindsey I; Frye, Stephen V.
Afiliação
  • Stuckey JI; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, USA.
  • Dickson BM; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, USA.
  • Cheng N; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, USA.
  • Liu Y; Structural Genomics Consortium, University of Toronto, Toronto, Ontario, Canada.
  • Norris JL; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, USA.
  • Cholensky SH; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, USA.
  • Tempel W; Structural Genomics Consortium, University of Toronto, Toronto, Ontario, Canada.
  • Qin S; Structural Genomics Consortium, University of Toronto, Toronto, Ontario, Canada.
  • Huber KG; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, USA.
  • Sagum C; Department of Epigenetics and Molecular Carcinogenesis, University of Texas MD Anderson Cancer Center, Smithville, Texas, USA.
  • Black K; Department of Epigenetics and Molecular Carcinogenesis, University of Texas MD Anderson Cancer Center, Smithville, Texas, USA.
  • Li F; Structural Genomics Consortium, University of Toronto, Toronto, Ontario, Canada.
  • Huang XP; National Institute of Mental Health Psychoactive Drug Screening Program, University of North Carolina at Chapel Hill Medical School, Chapel Hill, North Carolina, USA.
  • Roth BL; Department of Pharmacology, University of North Carolina at Chapel Hill Medical School, Chapel Hill, North Carolina, USA.
  • Baughman BM; National Institute of Mental Health Psychoactive Drug Screening Program, University of North Carolina at Chapel Hill Medical School, Chapel Hill, North Carolina, USA.
  • Senisterra G; Department of Pharmacology, University of North Carolina at Chapel Hill Medical School, Chapel Hill, North Carolina, USA.
  • Pattenden SG; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, USA.
  • Vedadi M; Structural Genomics Consortium, University of Toronto, Toronto, Ontario, Canada.
  • Brown PJ; Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina, USA.
  • Bedford MT; Structural Genomics Consortium, University of Toronto, Toronto, Ontario, Canada.
  • Min J; Structural Genomics Consortium, University of Toronto, Toronto, Ontario, Canada.
  • Arrowsmith CH; Department of Epigenetics and Molecular Carcinogenesis, University of Texas MD Anderson Cancer Center, Smithville, Texas, USA.
  • James LI; Structural Genomics Consortium, University of Toronto, Toronto, Ontario, Canada.
  • Frye SV; Structural Genomics Consortium, University of Toronto, Toronto, Ontario, Canada.
Nat Chem Biol ; 12(3): 180-7, 2016 Mar.
Article em En | MEDLINE | ID: mdl-26807715

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Oligopeptídeos / Complexo Repressor Polycomb 1 Limite: Animals / Humans / Male Idioma: En Revista: Nat Chem Biol Assunto da revista: BIOLOGIA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Oligopeptídeos / Complexo Repressor Polycomb 1 Limite: Animals / Humans / Male Idioma: En Revista: Nat Chem Biol Assunto da revista: BIOLOGIA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Estados Unidos