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Discovery of the ROCK inhibitor netarsudil for the treatment of open-angle glaucoma.
Sturdivant, Jill M; Royalty, Susan M; Lin, Cheng-Wen; Moore, Lori A; Yingling, Jeffrey D; Laethem, Carmen L; Sherman, Bryan; Heintzelman, Geoffrey R; Kopczynski, Casey C; deLong, Mitchell A.
Afiliação
  • Sturdivant JM; Aerie Pharmaceuticals, Inc., 4301 Emperor Boulevard, Suite 400, Durham, NC 27703, United States. Electronic address: jsturdivant@aeriepharma.com.
  • Royalty SM; Aerie Pharmaceuticals, Inc., 4301 Emperor Boulevard, Suite 400, Durham, NC 27703, United States.
  • Lin CW; Aerie Pharmaceuticals, Inc., 4301 Emperor Boulevard, Suite 400, Durham, NC 27703, United States.
  • Moore LA; Aerie Pharmaceuticals, Inc., 4301 Emperor Boulevard, Suite 400, Durham, NC 27703, United States.
  • Yingling JD; Aerie Pharmaceuticals, Inc., 4301 Emperor Boulevard, Suite 400, Durham, NC 27703, United States.
  • Laethem CL; Aerie Pharmaceuticals, Inc., 4301 Emperor Boulevard, Suite 400, Durham, NC 27703, United States.
  • Sherman B; Aerie Pharmaceuticals, Inc., 4301 Emperor Boulevard, Suite 400, Durham, NC 27703, United States.
  • Heintzelman GR; Aerie Pharmaceuticals, Inc., 4301 Emperor Boulevard, Suite 400, Durham, NC 27703, United States.
  • Kopczynski CC; Aerie Pharmaceuticals, Inc., 4301 Emperor Boulevard, Suite 400, Durham, NC 27703, United States.
  • deLong MA; Aerie Pharmaceuticals, Inc., 4301 Emperor Boulevard, Suite 400, Durham, NC 27703, United States.
Bioorg Med Chem Lett ; 26(10): 2475-2480, 2016 05 15.
Article em En | MEDLINE | ID: mdl-27072905

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Benzoatos / Glaucoma de Ângulo Aberto / Beta-Alanina / Inibidores de Proteínas Quinases / Quinases Associadas a rho Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Benzoatos / Glaucoma de Ângulo Aberto / Beta-Alanina / Inibidores de Proteínas Quinases / Quinases Associadas a rho Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article