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Discovery of Orally Efficacious Phosphoinositide 3-Kinase δ Inhibitors with Improved Metabolic Stability.
Patel, Leena; Chandrasekhar, Jayaraman; Evarts, Jerry; Forseth, Kristen; Haran, Aaron C; Ip, Carmen; Kashishian, Adam; Kim, Musong; Koditek, David; Koppenol, Sandy; Lad, Latesh; Lepist, Eve-Irene; McGrath, Mary E; Perreault, Stephane; Puri, Kamal D; Villaseñor, Armando G; Somoza, John R; Steiner, Bart H; Therrien, Joseph; Treiberg, Jennifer; Phillips, Gary.
Afiliação
  • Patel L; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Chandrasekhar J; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Evarts J; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Forseth K; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Haran AC; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Ip C; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Kashishian A; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Kim M; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Koditek D; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Koppenol S; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Lad L; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Lepist EI; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • McGrath ME; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Perreault S; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Puri KD; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Villaseñor AG; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Somoza JR; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Steiner BH; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Therrien J; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Treiberg J; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
  • Phillips G; Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, California 94404, United States.
J Med Chem ; 59(19): 9228-9242, 2016 Oct 13.
Article em En | MEDLINE | ID: mdl-27660855

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Estados Unidos