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C-Terminal residues in small potassium channel blockers OdK1 and OSK3 from scorpion venom fine-tune the selectivity.
Kuzmenkov, Alexey I; Peigneur, Steve; Chugunov, Anton O; Tabakmakher, Valentin M; Efremov, Roman G; Tytgat, Jan; Grishin, Eugene V; Vassilevski, Alexander A.
Afiliação
  • Kuzmenkov AI; Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow 117997, Russia; Biological Faculty, Lomonosov Moscow State University, Moscow 119992, Russia. Electronic address: aleksey.kuzmenkov@gmail.com.
  • Peigneur S; Toxicology and Pharmacology, University of Leuven, Leuven 3000, Belgium.
  • Chugunov AO; Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow 117997, Russia; National Research University Higher School of Economics, Moscow, 101000, Russia.
  • Tabakmakher VM; Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow 117997, Russia.
  • Efremov RG; Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow 117997, Russia; National Research University Higher School of Economics, Moscow, 101000, Russia.
  • Tytgat J; Toxicology and Pharmacology, University of Leuven, Leuven 3000, Belgium.
  • Grishin EV; Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow 117997, Russia.
  • Vassilevski AA; Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow 117997, Russia; Biological Faculty, Lomonosov Moscow State University, Moscow 119992, Russia. Electronic address: avas@ibch.ru.
Biochim Biophys Acta Proteins Proteom ; 1865(5): 465-472, 2017 May.
Article em En | MEDLINE | ID: mdl-28179135

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Conformação Proteica / Venenos de Escorpião / Bloqueadores dos Canais de Potássio Tipo de estudo: Prognostic_studies Limite: Animals Idioma: En Revista: Biochim Biophys Acta Proteins Proteom Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Conformação Proteica / Venenos de Escorpião / Bloqueadores dos Canais de Potássio Tipo de estudo: Prognostic_studies Limite: Animals Idioma: En Revista: Biochim Biophys Acta Proteins Proteom Ano de publicação: 2017 Tipo de documento: Article