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Uncialamycin as a novel payload for antibody drug conjugate (ADC) based targeted cancer therapy.
Chowdari, Naidu S; Pan, Chin; Rao, Chetana; Langley, David R; Sivaprakasam, Prasanna; Sufi, Bilal; Derwin, Daniel; Wang, Yichong; Kwok, Eilene; Passmore, David; Rangan, Vangipuram S; Deshpande, Shrikant; Cardarelli, Pina; Vite, Gregory; Gangwar, Sanjeev.
Afiliação
  • Chowdari NS; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA. Electronic address: naidu.chowdari@bms.com.
  • Pan C; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA.
  • Rao C; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA.
  • Langley DR; Bristol-Myers Squibb Research & Development, 5 Research Parkway, Wallingford, CT 06492, USA.
  • Sivaprakasam P; Bristol-Myers Squibb Research & Development, PO Box 4000, Princeton, NJ 08543, USA.
  • Sufi B; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA.
  • Derwin D; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA.
  • Wang Y; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA.
  • Kwok E; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA.
  • Passmore D; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA.
  • Rangan VS; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA.
  • Deshpande S; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA.
  • Cardarelli P; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA.
  • Vite G; Bristol-Myers Squibb Research & Development, PO Box 4000, Princeton, NJ 08543, USA.
  • Gangwar S; Bristol-Myers Squibb Research & Development, 700 Bay Road, Redwood City, CA 94063, USA.
Bioorg Med Chem Lett ; 29(3): 466-470, 2019 02 01.
Article em En | MEDLINE | ID: mdl-30579797

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antraquinonas / Imunoconjugados / Neoplasias Pulmonares / Anticorpos Monoclonais / Antineoplásicos Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antraquinonas / Imunoconjugados / Neoplasias Pulmonares / Anticorpos Monoclonais / Antineoplásicos Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2019 Tipo de documento: Article