ß-Arrestin-Biased AT1 Agonist TRV027 Causes a Neonatal-Specific Sustained Positive Inotropic Effect Without Increasing Heart Rate.
JACC Basic Transl Sci
; 5(11): 1057-1069, 2020 Nov.
Article
em En
| MEDLINE
| ID: mdl-33294739
AT1R, angiotensin type 1 receptor; AngII, angiotensin II; BBA, ß-arrestinbiased angiotensin type 1 receptor agonist; ECG, electrocardiography; GPCR, G proteincoupled receptor; LTCC, CaV1.2 L-type Ca2+ channel; OCR, oxygen consumption rate; PHF, pediatric heart failure; ROS, reactive oxygen species; TRV027; UCG, ultrasound cardiogram; congenital dilated cardiomyopathy; hiPSC-CM, human induced pluripotent stem cellderived cardiac myocyte; human induced pluripotent stem cell-derived cardiac myocytes; inotropic vasodilator; mNVCM, mouse neonatal ventricular cardiac myocyte; neonate; pediatric heart failure; ß-arrestinbiased AT1 angiotensin receptor agonist
Texto completo:
1
Coleções:
01-internacional
Base de dados:
MEDLINE
Tipo de estudo:
Etiology_studies
Idioma:
En
Revista:
JACC Basic Transl Sci
Ano de publicação:
2020
Tipo de documento:
Article
País de afiliação:
Japão