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Synthesis and Pharmacological Evaluation of Fluorinated Quinoxaline-Based κ-Opioid Receptor (KOR) Agonists Designed for PET Studies.
Tangherlini, Giovanni; Börgel, Frederik; Schepmann, Dirk; Slocum, Samuel; Che, Tao; Wagner, Stefan; Schwegmann, Katrin; Hermann, Sven; Mykicki, Nadine; Loser, Karin; Wünsch, Bernhard.
Afiliação
  • Tangherlini G; Institut für Pharmazeutische und Medizinische Chemie, Universität Münster, Corrensstraße 48, 48149, Münster, Germany.
  • Börgel F; Cells-in-Motion Cluster of Excellence (EXC 1003-CiM), Westfälische Wilhelms-Universität Münster, 48149, Münster, Germany.
  • Schepmann D; Institut für Pharmazeutische und Medizinische Chemie, Universität Münster, Corrensstraße 48, 48149, Münster, Germany.
  • Slocum S; Institut für Pharmazeutische und Medizinische Chemie, Universität Münster, Corrensstraße 48, 48149, Münster, Germany.
  • Che T; Department of Pharmacology, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, NC 27599, USA.
  • Wagner S; Department of Anesthesiology, Washington University School of Medicine, 660 S. Euclid Ave., St. Louis, MO 63110, USA.
  • Schwegmann K; Department of Nuclear Medicine, University Hospital Münster, Albert-Schweitzer-Campus 1, Building A1, 48149, Münster, Germany.
  • Hermann S; European Institute for Molecular Imaging (EIMI), University of Münster, Waldeyerstraße 15, 48149, Münster, Germany.
  • Mykicki N; European Institute for Molecular Imaging (EIMI), University of Münster, Waldeyerstraße 15, 48149, Münster, Germany.
  • Loser K; Department of Dermatology, University of Münster, von-Esmarch-Str. 58, 48149, Münster, Germany.
  • Wünsch B; Cells-in-Motion Cluster of Excellence (EXC 1003-CiM), Westfälische Wilhelms-Universität Münster, 48149, Münster, Germany.
ChemMedChem ; 15(19): 1834-1853, 2020 10 05.
Article em En | MEDLINE | ID: mdl-33448685

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinoxalinas / Anti-Inflamatórios não Esteroides / Receptores Opioides kappa / Compostos Radiofarmacêuticos Limite: Animals / Humans Idioma: En Revista: ChemMedChem Assunto da revista: FARMACOLOGIA / QUIMICA Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Alemanha

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinoxalinas / Anti-Inflamatórios não Esteroides / Receptores Opioides kappa / Compostos Radiofarmacêuticos Limite: Animals / Humans Idioma: En Revista: ChemMedChem Assunto da revista: FARMACOLOGIA / QUIMICA Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Alemanha