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A head-to-head comparison of the inhibitory activities of 15 peptidomimetic SARS-CoV-2 3CLpro inhibitors.
Vankadara, Subramanyam; Wong, Yun Xuan; Liu, Boping; See, Yi Yang; Tan, Li Hong; Tan, Qian Wen; Wang, Gang; Karuna, Ratna; Guo, Xue; Tan, Shu Ting; Fong, Jia Yi; Joy, Joma; Chia, C S Brian.
Afiliação
  • Vankadara S; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • Wong YX; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • Liu B; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • See YY; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • Tan LH; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • Tan QW; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • Wang G; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • Karuna R; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • Guo X; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • Tan ST; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • Fong JY; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • Joy J; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore.
  • Chia CSB; Experimental Drug Development Centre, 10 Biopolis Road, Chromos #08-01, Singapore 138670, Singapore. Electronic address: cschia@eddc.a-star.edu.sg.
Bioorg Med Chem Lett ; 48: 128263, 2021 09 15.
Article em En | MEDLINE | ID: mdl-34271072

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antivirais / Inibidores de Cisteína Proteinase / Peptidomiméticos / Proteases 3C de Coronavírus / SARS-CoV-2 Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Singapura

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antivirais / Inibidores de Cisteína Proteinase / Peptidomiméticos / Proteases 3C de Coronavírus / SARS-CoV-2 Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Singapura