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Structure-Activity Relationships of Triple-Action Platinum(IV) Prodrugs with Albumin-Binding Properties and Immunomodulating Ligands.
Fronik, Philipp; Poetsch, Isabella; Kastner, Alexander; Mendrina, Theresa; Hager, Sonja; Hohenwallner, Katharina; Schueffl, Hemma; Herndler-Brandstetter, Dietmar; Koellensperger, Gunda; Rampler, Evelyn; Kopecka, Joanna; Riganti, Chiara; Berger, Walter; Keppler, Bernhard K; Heffeter, Petra; Kowol, Christian R.
Afiliação
  • Fronik P; Faculty of Chemistry, Institute of Inorganic Chemistry, University of Vienna, Waehringer Strasse 42, 1090 Vienna, Austria.
  • Poetsch I; Faculty of Chemistry, Institute of Inorganic Chemistry, University of Vienna, Waehringer Strasse 42, 1090 Vienna, Austria.
  • Kastner A; Institute of Cancer Research and Comprehensive Cancer Center, Medical University of Vienna, Borschkegasse 8a, 1090 Vienna, Austria.
  • Mendrina T; Research Cluster "Translational Cancer Therapy Research", 1090 Vienna, Austria.
  • Hager S; Faculty of Chemistry, Institute of Inorganic Chemistry, University of Vienna, Waehringer Strasse 42, 1090 Vienna, Austria.
  • Hohenwallner K; Institute of Cancer Research and Comprehensive Cancer Center, Medical University of Vienna, Borschkegasse 8a, 1090 Vienna, Austria.
  • Schueffl H; Institute of Cancer Research and Comprehensive Cancer Center, Medical University of Vienna, Borschkegasse 8a, 1090 Vienna, Austria.
  • Herndler-Brandstetter D; Faculty of Chemistry, Institute of Analytical Chemistry, University of Vienna, Waehringer Strasse 38, 1090 Vienna, Austria.
  • Koellensperger G; Institute of Cancer Research and Comprehensive Cancer Center, Medical University of Vienna, Borschkegasse 8a, 1090 Vienna, Austria.
  • Rampler E; Institute of Cancer Research and Comprehensive Cancer Center, Medical University of Vienna, Borschkegasse 8a, 1090 Vienna, Austria.
  • Kopecka J; Faculty of Chemistry, Institute of Analytical Chemistry, University of Vienna, Waehringer Strasse 38, 1090 Vienna, Austria.
  • Riganti C; Faculty of Chemistry, Institute of Analytical Chemistry, University of Vienna, Waehringer Strasse 38, 1090 Vienna, Austria.
  • Berger W; Department of Oncology, University of Torino, via Santena 5/bis, 10126 Torino, Italy.
  • Keppler BK; Department of Oncology, University of Torino, via Santena 5/bis, 10126 Torino, Italy.
  • Heffeter P; Institute of Cancer Research and Comprehensive Cancer Center, Medical University of Vienna, Borschkegasse 8a, 1090 Vienna, Austria.
  • Kowol CR; Research Cluster "Translational Cancer Therapy Research", 1090 Vienna, Austria.
J Med Chem ; 64(16): 12132-12151, 2021 08 26.
Article em En | MEDLINE | ID: mdl-34403254

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pró-Fármacos / Complexos de Coordenação / Fatores Imunológicos / Maleimidas / Neoplasias / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Animals / Female / Humans / Male Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Áustria

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pró-Fármacos / Complexos de Coordenação / Fatores Imunológicos / Maleimidas / Neoplasias / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Animals / Female / Humans / Male Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Áustria