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Bioorg Med Chem Lett
; 18(19): 5263-7, 2008 Oct 01.
Artículo
en Inglés
| MEDLINE
| ID: mdl-18789686
RESUMEN
Novel 5,6-diarylimidazo[2,1-b][1,3]thiazoles bearing an amine substituent at the imidazothiazole 2-position have been synthesized and evaluated as anticoccidial agents in both in vitro and in vivo assays. Both subnanomolar in vitro activity and broad spectrum in vivo potency were detected for several compounds, particularly compound 10.