1.
Bioorg Med Chem Lett
; 20(9): 2968-73, 2010 May 01.
Artículo
en Inglés
| MEDLINE
| ID: mdl-20347591
RESUMEN
We describe the structure-activity relationship of the C1-group of pyrano[3,4-b]indole based inhibitors of HCV NS5B polymerase. Further exploration of the allosteric binding site led to the discovery of the significantly more potent compound 12.