1.
J Org Chem
; 75(24): 8670-3, 2010 Dec 17.
Artigo
em Inglês
| MEDLINE
| ID: mdl-21082772
RESUMO
Linear hydroformylation of N-protected allyl- or homoallylamines (cyclohydrocarbonylation: CHC), followed by a reductive amination constitute the two key steps toward convenient routes to aza-heterocycles.