NK1 antagonists based on seven membered lactam scaffolds.
Bioorg Med Chem Lett
; 16(11): 2929-32, 2006 Jun 01.
Article
en En
| MEDLINE
| ID: mdl-16574413
ABSTRACT
A new class of high affinity hNK1R antagonists based on seven-membered ring cores has been identified. This series, with relatively simple, compact structures, includes compounds with high affinity, good selectivity, and promising in vivo properties.
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Colección:
01-internacional
Banco de datos:
MEDLINE
Asunto principal:
Antagonistas del Receptor de Neuroquinina-1
/
Lactamas
Límite:
Humans
Idioma:
En
Revista:
Bioorg Med Chem Lett
Asunto de la revista:
BIOQUIMICA
/
QUIMICA
Año:
2006
Tipo del documento:
Article
País de afiliación:
Reino Unido