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Placement of Hydroxy Moiety on Pendant of Peptidomimetic Scaffold Modulates Mu and Kappa Opioid Receptor Efficacy.
Harland, Aubrie A; Pogozheva, Irina D; Griggs, Nicholas W; Trask, Tyler J; Traynor, John R; Mosberg, Henry I.
Afiliación
  • Harland AA; Department of Medicinal Chemistry, College of Pharmacy, University of Michigan , Ann Arbor, Michigan 48109, United States.
  • Pogozheva ID; Department of Medicinal Chemistry, College of Pharmacy, University of Michigan , Ann Arbor, Michigan 48109, United States.
  • Griggs NW; Department of Pharmacology, Medical School, University of Michigan , Ann Arbor, Michigan 48109, United States.
  • Trask TJ; Department of Pharmacology, Medical School, University of Michigan , Ann Arbor, Michigan 48109, United States.
  • Traynor JR; Department of Pharmacology, Medical School, University of Michigan , Ann Arbor, Michigan 48109, United States.
  • Mosberg HI; Department of Medicinal Chemistry, College of Pharmacy, University of Michigan , Ann Arbor, Michigan 48109, United States.
ACS Chem Neurosci ; 8(11): 2549-2557, 2017 11 15.
Article en En | MEDLINE | ID: mdl-28796483

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Receptores Opioides delta / Receptores Opioides kappa / Receptores Opioides mu / Peptidomiméticos / Analgésicos Opioides Límite: Animals / Humans Idioma: En Revista: ACS Chem Neurosci Año: 2017 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Receptores Opioides delta / Receptores Opioides kappa / Receptores Opioides mu / Peptidomiméticos / Analgésicos Opioides Límite: Animals / Humans Idioma: En Revista: ACS Chem Neurosci Año: 2017 Tipo del documento: Article País de afiliación: Estados Unidos