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C-H Arylation in the Formation of a Complex Pyrrolopyridine, the Commercial Synthesis of the Potent JAK2 Inhibitor, BMS-911543.
Fox, Richard J; Cuniere, Nicolas L; Bakrania, Lopa; Wei, Carolyn; Strotman, Neil A; Hay, Michael; Fanfair, Dayne; Regens, Christopher; Beutner, Gregory L; Lawler, Michael; Lobben, Paul; Soumeillant, Maxime C; Cohen, Benjamin; Zhu, Keming; Skliar, Dimitri; Rosner, Thorsten; Markwalter, Chester E; Hsiao, Yi; Tran, Kristy; Eastgate, Martin D.
Afiliación
  • Fox RJ; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Cuniere NL; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Bakrania L; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Wei C; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Strotman NA; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Hay M; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Fanfair D; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Regens C; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Beutner GL; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Lawler M; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Lobben P; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Soumeillant MC; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Cohen B; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Zhu K; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Skliar D; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Rosner T; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Markwalter CE; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Hsiao Y; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Tran K; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
  • Eastgate MD; Chemical Development , Bristol-Myers Squibb , One Squibb Drive , New Brunswick , New Jersey 08903 , United States.
J Org Chem ; 84(8): 4661-4669, 2019 04 19.
Article en En | MEDLINE | ID: mdl-30388009

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Inhibidores de Proteínas Quinasas / Compuestos Heterocíclicos con 3 Anillos Límite: Humans Idioma: En Revista: J Org Chem Año: 2019 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Inhibidores de Proteínas Quinasas / Compuestos Heterocíclicos con 3 Anillos Límite: Humans Idioma: En Revista: J Org Chem Año: 2019 Tipo del documento: Article País de afiliación: Estados Unidos