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Optimization of substituted cinnamic acyl sulfonamide derivatives as tubulin polymerization inhibitors with anticancer activity.
Luo, Yin; Zhou, Yang; Song, Yanhua; Chen, Guo; Wang, Yu-Xiang; Tian, Ye; Fan, Wei-Wei; Yang, Yu-Shun; Cheng, Tao; Zhu, Hai-Liang.
Afiliación
  • Luo Y; Department of Neurosurgery, Changhai Hospital, Second Military Medical University, Shanghai 200433, People's Republic of China. Electronic address: luoyin147@163.com.
  • Zhou Y; Cixi Institute of BioMedical Engineering, Ningbo Institute of Industrial Technology, CAS, Ningbo 315201, People's Republic of China.
  • Song Y; Tianjin 4th Centre Hospital, Tianjin 300140, People's Republic of China.
  • Chen G; Department of Radiation Oncology, Emory University School of Medicine and Winship Cancer Institute of Emory University, Atlanta, GA 30322, USA.
  • Wang YX; State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, People's Republic of China.
  • Tian Y; State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, People's Republic of China.
  • Fan WW; State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, People's Republic of China.
  • Yang YS; State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, People's Republic of China.
  • Cheng T; Pharmaron Ningbo Co., Ltd., Ningbo 315366,People's Republic of China.
  • Zhu HL; State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, People's Republic of China. Electronic address: zhuhl@nju.edu.cn.
Bioorg Med Chem Lett ; 28(23-24): 3634-3638, 2018 12 15.
Article en En | MEDLINE | ID: mdl-30389289

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Sulfonamidas / Tubulina (Proteína) / Moduladores de Tubulina Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2018 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Sulfonamidas / Tubulina (Proteína) / Moduladores de Tubulina Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2018 Tipo del documento: Article