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Implementation of the CYP Index for the Design of Selective Tryptophan-2,3-dioxygenase Inhibitors.
Parr, Brendan T; Pastor, Richard; Sellers, Benjamin D; Pei, Zhonghua; Jaipuri, Firoz A; Castanedo, Georgette M; Gazzard, Lewis; Kumar, Sanjeev; Li, Xiaokai; Liu, Wen; Mendonca, Rohan; Pavana, Roheeth K; Potturi, Hima; Shao, Cheng; Velvadapu, Venkata; Waldo, Jesse P; Wu, Guosheng; Yuen, Po-Wai; Zhang, Zuhui; Zhang, Yamin; Harris, Seth F; Oh, Angela J; DiPasquale, Antonio; Dement, Kevin; La, Hank; Goon, Leanne; Gustafson, Amy; VanderPorten, Erica C; Mautino, Mario R; Liu, Yichin.
Afiliación
  • Parr BT; Genentech, South San Francisco, California 94080, United States.
  • Pastor R; Genentech, South San Francisco, California 94080, United States.
  • Sellers BD; Genentech, South San Francisco, California 94080, United States.
  • Pei Z; Genentech, South San Francisco, California 94080, United States.
  • Jaipuri FA; NewLink Genetics, Ames, Iowa 50010, United States.
  • Castanedo GM; Genentech, South San Francisco, California 94080, United States.
  • Gazzard L; Genentech, South San Francisco, California 94080, United States.
  • Kumar S; NewLink Genetics, Ames, Iowa 50010, United States.
  • Li X; NewLink Genetics, Ames, Iowa 50010, United States.
  • Liu W; Genentech, South San Francisco, California 94080, United States.
  • Mendonca R; Genentech, South San Francisco, California 94080, United States.
  • Pavana RK; NewLink Genetics, Ames, Iowa 50010, United States.
  • Potturi H; NewLink Genetics, Ames, Iowa 50010, United States.
  • Shao C; Pharmaron, Beijing 100176, People's Republic of China.
  • Velvadapu V; NewLink Genetics, Ames, Iowa 50010, United States.
  • Waldo JP; NewLink Genetics, Ames, Iowa 50010, United States.
  • Wu G; Pharmaron, Beijing 100176, People's Republic of China.
  • Yuen PW; Pharmaron, Beijing 100176, People's Republic of China.
  • Zhang Z; NewLink Genetics, Ames, Iowa 50010, United States.
  • Zhang Y; Pharmaron, Beijing 100176, People's Republic of China.
  • Harris SF; Genentech, South San Francisco, California 94080, United States.
  • Oh AJ; Genentech, South San Francisco, California 94080, United States.
  • DiPasquale A; Genentech, South San Francisco, California 94080, United States.
  • Dement K; Genentech, South San Francisco, California 94080, United States.
  • La H; Genentech, South San Francisco, California 94080, United States.
  • Goon L; Genentech, South San Francisco, California 94080, United States.
  • Gustafson A; Genentech, South San Francisco, California 94080, United States.
  • VanderPorten EC; Genentech, South San Francisco, California 94080, United States.
  • Mautino MR; NewLink Genetics, Ames, Iowa 50010, United States.
  • Liu Y; Genentech, South San Francisco, California 94080, United States.
ACS Med Chem Lett ; 11(4): 541-549, 2020 Apr 09.
Article en En | MEDLINE | ID: mdl-32292562

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos