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Allosteric Inhibition of the SARS-CoV-2 Main Protease: Insights from Mass Spectrometry Based Assays*.
El-Baba, Tarick J; Lutomski, Corinne A; Kantsadi, Anastassia L; Malla, Tika R; John, Tobias; Mikhailov, Victor; Bolla, Jani R; Schofield, Christopher J; Zitzmann, Nicole; Vakonakis, Ioannis; Robinson, Carol V.
Afiliación
  • El-Baba TJ; Physical and Theoretical Chemistry Laboratory, University of Oxford, South Parks Rd., OX1 3QZ, Oxford, UK.
  • Lutomski CA; Physical and Theoretical Chemistry Laboratory, University of Oxford, South Parks Rd., OX1 3QZ, Oxford, UK.
  • Kantsadi AL; Department of Biochemistry, University of Oxford, South Parks Rd., OX1 3QU, Oxford, UK.
  • Malla TR; Chemistry Research Laboratory, University of Oxford, 12 Mansfield Rd, OX1 3TA, Oxford, UK.
  • John T; Chemistry Research Laboratory, University of Oxford, 12 Mansfield Rd, OX1 3TA, Oxford, UK.
  • Mikhailov V; Chemistry Research Laboratory, University of Oxford, 12 Mansfield Rd, OX1 3TA, Oxford, UK.
  • Bolla JR; Physical and Theoretical Chemistry Laboratory, University of Oxford, South Parks Rd., OX1 3QZ, Oxford, UK.
  • Schofield CJ; Chemistry Research Laboratory, University of Oxford, 12 Mansfield Rd, OX1 3TA, Oxford, UK.
  • Zitzmann N; Department of Biochemistry, University of Oxford, South Parks Rd., OX1 3QU, Oxford, UK.
  • Vakonakis I; Department of Biochemistry, University of Oxford, South Parks Rd., OX1 3QU, Oxford, UK.
  • Robinson CV; Physical and Theoretical Chemistry Laboratory, University of Oxford, South Parks Rd., OX1 3QZ, Oxford, UK.
Angew Chem Int Ed Engl ; 59(52): 23544-23548, 2020 12 21.
Article en En | MEDLINE | ID: mdl-32841477

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Modelos Moleculares / Bibliotecas de Moléculas Pequeñas / Inhibidores de Proteasa de Coronavirus / Proteasas 3C de Coronavirus / SARS-CoV-2 Idioma: En Revista: Angew Chem Int Ed Engl Año: 2020 Tipo del documento: Article País de afiliación: Reino Unido

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Modelos Moleculares / Bibliotecas de Moléculas Pequeñas / Inhibidores de Proteasa de Coronavirus / Proteasas 3C de Coronavirus / SARS-CoV-2 Idioma: En Revista: Angew Chem Int Ed Engl Año: 2020 Tipo del documento: Article País de afiliación: Reino Unido