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Simultaneous CK2/TNIK/DYRK1 inhibition by 108600 suppresses triple negative breast cancer stem cells and chemotherapy-resistant disease.
Sato, Katsutoshi; Padgaonkar, Amol A; Baker, Stacey J; Cosenza, Stephen C; Rechkoblit, Olga; Subbaiah, D R C Venkata; Domingo-Domenech, Josep; Bartkowski, Alison; Port, Elisa R; Aggarwal, Aneel K; Ramana Reddy, M V; Irie, Hanna Y; Reddy, E Premkumar.
Afiliación
  • Sato K; Division of Hematology and Medical Oncology, Department of Medicine, Icahn School of Medicine at Mount Sinai, New York, NY, USA.
  • Padgaonkar AA; Department of Oncological Sciences, Icahn School of Medicine at Mount Sinai, New York, NY, USA.
  • Baker SJ; Department of Oncological Sciences, Icahn School of Medicine at Mount Sinai, New York, NY, USA.
  • Cosenza SC; Department of Oncological Sciences, Icahn School of Medicine at Mount Sinai, New York, NY, USA.
  • Rechkoblit O; Department of Pharmacological Sciences, Icahn School of Medicine at Mount Sinai, New York, NY, USA.
  • Subbaiah DRCV; Department of Oncological Sciences, Icahn School of Medicine at Mount Sinai, New York, NY, USA.
  • Domingo-Domenech J; Medical Oncology and Cancer Biology, Thomas Jefferson University, Philadelphia, PA, USA.
  • Bartkowski A; Division of Hematology and Medical Oncology, Department of Medicine, Icahn School of Medicine at Mount Sinai, New York, NY, USA.
  • Port ER; Department of Surgery, Mount Sinai Hospital, New York, NY, USA.
  • Aggarwal AK; Department of Pharmacological Sciences, Icahn School of Medicine at Mount Sinai, New York, NY, USA.
  • Ramana Reddy MV; Department of Oncological Sciences, Icahn School of Medicine at Mount Sinai, New York, NY, USA.
  • Irie HY; Division of Hematology and Medical Oncology, Department of Medicine, Icahn School of Medicine at Mount Sinai, New York, NY, USA. hanna.irie@mssm.edu.
  • Reddy EP; Department of Oncological Sciences, Icahn School of Medicine at Mount Sinai, New York, NY, USA. hanna.irie@mssm.edu.
Nat Commun ; 12(1): 4671, 2021 08 03.
Article en En | MEDLINE | ID: mdl-34344863

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Tiazinas / Células Madre Neoplásicas / Protocolos de Quimioterapia Combinada Antineoplásica / Resistencia a Antineoplásicos / Inhibidores de Proteínas Quinasas / Neoplasias de la Mama Triple Negativas / Nitrobencenos Límite: Animals / Humans Idioma: En Revista: Nat Commun Asunto de la revista: BIOLOGIA / CIENCIA Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Tiazinas / Células Madre Neoplásicas / Protocolos de Quimioterapia Combinada Antineoplásica / Resistencia a Antineoplásicos / Inhibidores de Proteínas Quinasas / Neoplasias de la Mama Triple Negativas / Nitrobencenos Límite: Animals / Humans Idioma: En Revista: Nat Commun Asunto de la revista: BIOLOGIA / CIENCIA Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos