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Substrate-Inspired Fragment Merging and Growing Affords Efficacious LasB Inhibitors.
Kaya, Cansu; Walter, Isabell; Yahiaoui, Samir; Sikandar, Asfandyar; Alhayek, Alaa; Konstantinovic, Jelena; Kany, Andreas M; Haupenthal, Jörg; Köhnke, Jesko; Hartmann, Rolf W; Hirsch, Anna K H.
Afiliación
  • Kaya C; Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), Helmholtz Centre for Infection Research (HZI), Campus E8.1, 66123, Saarbrücken, Germany.
  • Walter I; Department of Pharmacy, Saarland University, Campus E8.1, 66123, Saarbrücken, Germany.
  • Yahiaoui S; Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), Helmholtz Centre for Infection Research (HZI), Campus E8.1, 66123, Saarbrücken, Germany.
  • Sikandar A; Department of Pharmacy, Saarland University, Campus E8.1, 66123, Saarbrücken, Germany.
  • Alhayek A; Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), Helmholtz Centre for Infection Research (HZI), Campus E8.1, 66123, Saarbrücken, Germany.
  • Konstantinovic J; Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), Helmholtz Centre for Infection Research (HZI), Campus E8.1, 66123, Saarbrücken, Germany.
  • Kany AM; Department of Pharmacy, Saarland University, Campus E8.1, 66123, Saarbrücken, Germany.
  • Haupenthal J; Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), Helmholtz Centre for Infection Research (HZI), Campus E8.1, 66123, Saarbrücken, Germany.
  • Köhnke J; Department of Pharmacy, Saarland University, Campus E8.1, 66123, Saarbrücken, Germany.
  • Hartmann RW; Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), Helmholtz Centre for Infection Research (HZI), Campus E8.1, 66123, Saarbrücken, Germany.
  • Hirsch AKH; Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), Helmholtz Centre for Infection Research (HZI), Campus E8.1, 66123, Saarbrücken, Germany.
Angew Chem Int Ed Engl ; 61(5): e202112295, 2022 01 26.
Article en En | MEDLINE | ID: mdl-34762767

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Pseudomonas aeruginosa Idioma: En Revista: Angew Chem Int Ed Engl Año: 2022 Tipo del documento: Article País de afiliación: Alemania

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Pseudomonas aeruginosa Idioma: En Revista: Angew Chem Int Ed Engl Año: 2022 Tipo del documento: Article País de afiliación: Alemania