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Structure-based discovery of conformationally selective inhibitors of the serotonin transporter.
Singh, Isha; Seth, Anubha; Billesbølle, Christian B; Braz, Joao; Rodriguiz, Ramona M; Roy, Kasturi; Bekele, Bethlehem; Craik, Veronica; Huang, Xi-Ping; Boytsov, Danila; Pogorelov, Vladimir M; Lak, Parnian; O'Donnell, Henry; Sandtner, Walter; Irwin, John J; Roth, Bryan L; Basbaum, Allan I; Wetsel, William C; Manglik, Aashish; Shoichet, Brian K; Rudnick, Gary.
Afiliación
  • Singh I; Department of Pharmaceutical Chemistry, University of California, San Francisco, 1700 4th St., Byers Hall Suite 508D, San Francisco, CA 94143, USA.
  • Seth A; Department of Pharmacology, Yale University School of Medicine, 333 Cedar Street, New Haven, CT 06520-8066, USA.
  • Billesbølle CB; Department of Pharmaceutical Chemistry, University of California, San Francisco, 1700 4th St., Byers Hall Suite 508D, San Francisco, CA 94143, USA.
  • Braz J; Department of Anatomy, University of California, San Francisco, San Francisco, CA 94143, USA.
  • Rodriguiz RM; Department of Psychiatry and Behavioral Sciences, Duke University Medical Center, Durham, NC 27710, USA; Mouse Behavioral and Neuroendocrine Analysis Core Facility, Duke University Medical Center, Durham, NC 27710, USA.
  • Roy K; Department of Pharmacology, Yale University School of Medicine, 333 Cedar Street, New Haven, CT 06520-8066, USA.
  • Bekele B; Department of Pharmacology, Yale University School of Medicine, 333 Cedar Street, New Haven, CT 06520-8066, USA.
  • Craik V; Department of Anatomy, University of California, San Francisco, San Francisco, CA 94143, USA.
  • Huang XP; Department of Pharmacology, NIMH Psychoactive Drug Screening Program, School of Medicine, University of North Carolina at Chapel Hill, Chapel Hill, NC 27599, USA.
  • Boytsov D; Institute of Pharmacology, Center for Physiology and Pharmacology, Medical University of Vienna, 1090 Vienna, Austria.
  • Pogorelov VM; Department of Psychiatry and Behavioral Sciences, Duke University Medical Center, Durham, NC 27710, USA.
  • Lak P; Department of Pharmaceutical Chemistry, University of California, San Francisco, 1700 4th St., Byers Hall Suite 508D, San Francisco, CA 94143, USA.
  • O'Donnell H; Department of Pharmaceutical Chemistry, University of California, San Francisco, 1700 4th St., Byers Hall Suite 508D, San Francisco, CA 94143, USA.
  • Sandtner W; Institute of Pharmacology, Center for Physiology and Pharmacology, Medical University of Vienna, 1090 Vienna, Austria.
  • Irwin JJ; Department of Pharmaceutical Chemistry, University of California, San Francisco, 1700 4th St., Byers Hall Suite 508D, San Francisco, CA 94143, USA.
  • Roth BL; Department of Pharmacology, NIMH Psychoactive Drug Screening Program, School of Medicine, University of North Carolina at Chapel Hill, Chapel Hill, NC 27599, USA; Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hi
  • Basbaum AI; Department of Anatomy, University of California, San Francisco, San Francisco, CA 94143, USA. Electronic address: allan.basbaum@ucsf.edu.
  • Wetsel WC; Department of Psychiatry and Behavioral Sciences, Duke University Medical Center, Durham, NC 27710, USA; Mouse Behavioral and Neuroendocrine Analysis Core Facility, Duke University Medical Center, Durham, NC 27710, USA; Departments of Cell Biology and Neurobiology, Duke University Medical Center, Du
  • Manglik A; Department of Pharmaceutical Chemistry, University of California, San Francisco, 1700 4th St., Byers Hall Suite 508D, San Francisco, CA 94143, USA; Department of Anesthesia and Perioperative Care, University of California, San Francisco, San Francisco, CA 94115, USA. Electronic address: aashish.mang
  • Shoichet BK; Department of Pharmaceutical Chemistry, University of California, San Francisco, 1700 4th St., Byers Hall Suite 508D, San Francisco, CA 94143, USA. Electronic address: bshoichet@gmail.com.
  • Rudnick G; Department of Pharmacology, Yale University School of Medicine, 333 Cedar Street, New Haven, CT 06520-8066, USA. Electronic address: gary.rudnick@yale.edu.
Cell ; 186(10): 2160-2175.e17, 2023 05 11.
Article en En | MEDLINE | ID: mdl-37137306

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Inhibidores Selectivos de la Recaptación de Serotonina / Proteínas de Transporte de Serotonina en la Membrana Plasmática / Bibliotecas de Moléculas Pequeñas / Ibogaína Límite: Animals Idioma: En Revista: Cell Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Inhibidores Selectivos de la Recaptación de Serotonina / Proteínas de Transporte de Serotonina en la Membrana Plasmática / Bibliotecas de Moléculas Pequeñas / Ibogaína Límite: Animals Idioma: En Revista: Cell Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos