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Design, synthesis, activity and molecular dynamics studies of 1,3,4-thiadiazole derivatives as selective allosteric inhibitors of SHP2 for the treatment of cancer.
Liu, Wen-Shan; Zhao, Ji-Feng; Guo, Xiao-Jing; Lu, Sheng-Ze; Li, Wei; Li, Wan-Zhong.
Afiliación
  • Liu WS; Shandong Key Laboratory of Medicine and Health (Clinical Applied Pharmacology), Department of Pharmacy, Affiliated Hospital of Weifang Medical University, Weifang, 261041, Shandong Province, China; Clinical Research Center, Affiliated Hospital of Weifang Medical University, Weifang, 261041, Shandong
  • Zhao JF; Shandong Key Laboratory of Medicine and Health (Clinical Applied Pharmacology), Department of Pharmacy, Affiliated Hospital of Weifang Medical University, Weifang, 261041, Shandong Province, China; Clinical Research Center, Affiliated Hospital of Weifang Medical University, Weifang, 261041, Shandong
  • Guo XJ; Clinical Research Center, Affiliated Hospital of Weifang Medical University, Weifang, 261041, Shandong Province, China.
  • Lu SZ; School of Pharmacy, Weifang Medical University, Weifang, 261053, Shandong Province, China.
  • Li W; School of Pharmacy, Weifang Medical University, Weifang, 261053, Shandong Province, China.
  • Li WZ; School of Pharmacy, Weifang Medical University, Weifang, 261053, Shandong Province, China. Electronic address: liwz@wfmc.edu.cn.
Eur J Med Chem ; 258: 115585, 2023 Oct 05.
Article en En | MEDLINE | ID: mdl-37390510

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Tiadiazoles / Neoplasias Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2023 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Tiadiazoles / Neoplasias Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2023 Tipo del documento: Article