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Discovery of SOAT2 inhibitors from synthetic small molecules.
Kobayashi, Keisuke; Ohshiro, Taichi; Tomoda, Hiroshi; Yin, Feng; Cui, Hai-Lei; Chouthaiwale, Pandurang V; Tanaka, Fujie.
Afiliação
  • Kobayashi K; Graduate School of Pharmaceutical Sciences, Kitasato University, 5-9-1 Shirokane, Minato-ku, Tokyo 108-8641, Japan.
  • Ohshiro T; Graduate School of Pharmaceutical Sciences, Kitasato University, 5-9-1 Shirokane, Minato-ku, Tokyo 108-8641, Japan.
  • Tomoda H; Graduate School of Pharmaceutical Sciences, Kitasato University, 5-9-1 Shirokane, Minato-ku, Tokyo 108-8641, Japan. Electronic address: tomodah@pharm.kitasato-u.ac.jp.
  • Yin F; Chemistry and Chemical Bioengineering Unit, Okinawa Institute of Science and Technology Graduate University, 1919-1 Tancha, Onna, Okinawa 904-0495, Japan.
  • Cui HL; Chemistry and Chemical Bioengineering Unit, Okinawa Institute of Science and Technology Graduate University, 1919-1 Tancha, Onna, Okinawa 904-0495, Japan.
  • Chouthaiwale PV; Chemistry and Chemical Bioengineering Unit, Okinawa Institute of Science and Technology Graduate University, 1919-1 Tancha, Onna, Okinawa 904-0495, Japan.
  • Tanaka F; Chemistry and Chemical Bioengineering Unit, Okinawa Institute of Science and Technology Graduate University, 1919-1 Tancha, Onna, Okinawa 904-0495, Japan. Electronic address: ftanaka@oist.jp.
Bioorg Med Chem Lett ; 26(24): 5899-5901, 2016 Dec 15.
Article em En | MEDLINE | ID: mdl-27876317

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piranos / Esterol O-Aciltransferase / Inibidores Enzimáticos / Bibliotecas de Moléculas Pequenas / Descoberta de Drogas Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Japão

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piranos / Esterol O-Aciltransferase / Inibidores Enzimáticos / Bibliotecas de Moléculas Pequenas / Descoberta de Drogas Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Japão