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Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform.
Moraes, Carolina B; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Calogeropoulou, Theodora; Prousis, Kyriakos C; Mangani, Stefano; Di Pisa, Flavio; Landi, Giacomo; Iacono, Lucia Dello; Pozzi, Cecilia; Freitas-Junior, Lucio H; Dos Santos Pascoalino, Bruno; Bertolacini, Claudia P; Behrens, Birte; Keminer, Oliver; Leu, Jennifer; Wolf, Markus; Reinshagen, Jeanette; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Venturelli, Alberto; Wrigley, Stephen; Karunakaran, Deepa; Kebede, Bethlehem; Pöhner, Ina; Müller, Wolfgang; Panecka-Hofman, Joanna; Wade, Rebecca C; Fenske, Martina; Clos, Joachim; Alunda, José María; Corral, María Jesús; Uliassi, Elisa; Bolognesi, Maria Laura; Linciano, Pasquale; Quotadamo, Antonio; Ferrari, Stefania; Santucci, Matteo; Borsari, Chiara; Costi, Maria Paola; Gul, Sheraz.
Afiliação
  • Moraes CB; 1 Laboratório Nacional de Biociências (LNBio), Centro de Pesquisa em Energia e Materiais (CNPEM), Campinas-SP, Brazil.
  • Witt G; 2 Department of Microbiology, Institute of Biomedical Sciences, University of São Paulo, São Paulo-SP, Brazil.
  • Kuzikov M; 3 Fraunhofer Institute for Molecular Biology and Applied Ecology-ScreeningPort, Hamburg, Germany.
  • Ellinger B; 3 Fraunhofer Institute for Molecular Biology and Applied Ecology-ScreeningPort, Hamburg, Germany.
  • Calogeropoulou T; 3 Fraunhofer Institute for Molecular Biology and Applied Ecology-ScreeningPort, Hamburg, Germany.
  • Prousis KC; 4 National Hellenic Research Foundation, Institute of Biology, Medicinal Chemistry and Biotechnology, Athens, Greece.
  • Mangani S; 4 National Hellenic Research Foundation, Institute of Biology, Medicinal Chemistry and Biotechnology, Athens, Greece.
  • Di Pisa F; 5 Department of Biotechnology, Chemistry and Pharmacy, University of Siena, Siena, Italy.
  • Landi G; 5 Department of Biotechnology, Chemistry and Pharmacy, University of Siena, Siena, Italy.
  • Iacono LD; 5 Department of Biotechnology, Chemistry and Pharmacy, University of Siena, Siena, Italy.
  • Pozzi C; 5 Department of Biotechnology, Chemistry and Pharmacy, University of Siena, Siena, Italy.
  • Freitas-Junior LH; 5 Department of Biotechnology, Chemistry and Pharmacy, University of Siena, Siena, Italy.
  • Dos Santos Pascoalino B; 1 Laboratório Nacional de Biociências (LNBio), Centro de Pesquisa em Energia e Materiais (CNPEM), Campinas-SP, Brazil.
  • Bertolacini CP; 2 Department of Microbiology, Institute of Biomedical Sciences, University of São Paulo, São Paulo-SP, Brazil.
  • Behrens B; 1 Laboratório Nacional de Biociências (LNBio), Centro de Pesquisa em Energia e Materiais (CNPEM), Campinas-SP, Brazil.
  • Keminer O; 1 Laboratório Nacional de Biociências (LNBio), Centro de Pesquisa em Energia e Materiais (CNPEM), Campinas-SP, Brazil.
  • Leu J; 3 Fraunhofer Institute for Molecular Biology and Applied Ecology-ScreeningPort, Hamburg, Germany.
  • Wolf M; 3 Fraunhofer Institute for Molecular Biology and Applied Ecology-ScreeningPort, Hamburg, Germany.
  • Reinshagen J; 3 Fraunhofer Institute for Molecular Biology and Applied Ecology-ScreeningPort, Hamburg, Germany.
  • Cordeiro-da-Silva A; 3 Fraunhofer Institute for Molecular Biology and Applied Ecology-ScreeningPort, Hamburg, Germany.
  • Santarem N; 3 Fraunhofer Institute for Molecular Biology and Applied Ecology-ScreeningPort, Hamburg, Germany.
  • Venturelli A; 6 Instituto de Investigação e Inovação em Saúde, Universidade do Porto and Institute for Molecular and Cell Biology, Porto, Portugal.
  • Wrigley S; 6 Instituto de Investigação e Inovação em Saúde, Universidade do Porto and Institute for Molecular and Cell Biology, Porto, Portugal.
  • Karunakaran D; 7 Tydock Pharma srl, Modena, Italy.
  • Kebede B; 8 Hypha Discovery Ltd, Slough, UK.
  • Pöhner I; 8 Hypha Discovery Ltd, Slough, UK.
  • Müller W; 8 Hypha Discovery Ltd, Slough, UK.
  • Panecka-Hofman J; 9 Molecular and Cellular Modeling Group, Heidelberg Institute for Theoretical Studies, Heidelberg, Germany.
  • Wade RC; 9 Molecular and Cellular Modeling Group, Heidelberg Institute for Theoretical Studies, Heidelberg, Germany.
  • Fenske M; 9 Molecular and Cellular Modeling Group, Heidelberg Institute for Theoretical Studies, Heidelberg, Germany.
  • Clos J; 11 Faculty of Physics, University of Warsaw, Warsaw, Poland.
  • Alunda JM; 9 Molecular and Cellular Modeling Group, Heidelberg Institute for Theoretical Studies, Heidelberg, Germany.
  • Corral MJ; 12 Center for Molecular Biology (ZMBH), DKFZ-ZMBH Alliance, Heidelberg University, Heidelberg, Germany.
  • Uliassi E; 13 Interdisciplinary Center for Scientific Computing (IWR), Heidelberg University, Heidelberg, Germany.
  • Bolognesi ML; 14 Fraunhofer Institute for Molecular Biology and Applied Ecology IME, Aachen, Germany.
  • Linciano P; 15 Bernhard Nocht Institute for Tropical Medicine, Hamburg, Germany.
  • Quotadamo A; 16 Complutense University of Madrid, Madrid, Spain.
  • Ferrari S; 16 Complutense University of Madrid, Madrid, Spain.
  • Santucci M; 17 Department of Pharmacy and Biotechnology, University of Bologna, Bologna, Italy.
  • Borsari C; 17 Department of Pharmacy and Biotechnology, University of Bologna, Bologna, Italy.
  • Costi MP; 18 Department of Life Sciences, University of Modena and Reggio Emilia, Modena, Italy.
  • Gul S; 18 Department of Life Sciences, University of Modena and Reggio Emilia, Modena, Italy.
SLAS Discov ; 24(3): 346-361, 2019 03.
Article em En | MEDLINE | ID: mdl-30784368

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Tripanossomicidas / Tripanossomíase / Descoberta de Drogas Limite: Humans Idioma: En Revista: SLAS Discov Ano de publicação: 2019 Tipo de documento: Article País de afiliação: Brasil

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Tripanossomicidas / Tripanossomíase / Descoberta de Drogas Limite: Humans Idioma: En Revista: SLAS Discov Ano de publicação: 2019 Tipo de documento: Article País de afiliação: Brasil