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Synthesis of analogs of the Gwt1 inhibitor manogepix (APX001A) and in vitro evaluation against Cryptococcus spp.
Trzoss, Michael; Covel, Jonathan A; Kapoor, Mili; Moloney, Molly K; Soltow, Quinlyn A; Webb, Peter J; Shaw, Karen Joy.
Afiliação
  • Trzoss M; Amplyx Pharmaceuticals, 12730 High Bluff Dr #160, San Diego, CA 92130, United States. Electronic address: trzossmichael@gmail.com.
  • Covel JA; Amplyx Pharmaceuticals, 12730 High Bluff Dr #160, San Diego, CA 92130, United States.
  • Kapoor M; Amplyx Pharmaceuticals, 12730 High Bluff Dr #160, San Diego, CA 92130, United States.
  • Moloney MK; Amplyx Pharmaceuticals, 12730 High Bluff Dr #160, San Diego, CA 92130, United States.
  • Soltow QA; Amplyx Pharmaceuticals, 12730 High Bluff Dr #160, San Diego, CA 92130, United States.
  • Webb PJ; Amplyx Pharmaceuticals, 12730 High Bluff Dr #160, San Diego, CA 92130, United States.
  • Shaw KJ; Amplyx Pharmaceuticals, 12730 High Bluff Dr #160, San Diego, CA 92130, United States. Electronic address: kshaw@amplyx.com.
Bioorg Med Chem Lett ; 29(23): 126713, 2019 12 01.
Article em En | MEDLINE | ID: mdl-31668974

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Cryptococcus / Proteínas de Saccharomyces cerevisiae / Aminopiridinas / Isoxazóis / Antifúngicos Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Cryptococcus / Proteínas de Saccharomyces cerevisiae / Aminopiridinas / Isoxazóis / Antifúngicos Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2019 Tipo de documento: Article