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A Benzodiazepine Ligand with Improved GABAA Receptor α5-Subunit Selectivity Driven by Interactions with Loop C.
Simeone, Xenia; Koniuszewski, Filip; Müllegger, Markus; Smetka, Andreas; Steudle, Friederike; Puthenkalam, Roshan; Ernst, Margot; Scholze, Petra.
Afiliação
  • Simeone X; Center for Brain Research, Medical University of Vienna, Vienna, Austria.
  • Koniuszewski F; Center for Brain Research, Medical University of Vienna, Vienna, Austria.
  • Müllegger M; Center for Brain Research, Medical University of Vienna, Vienna, Austria.
  • Smetka A; Center for Brain Research, Medical University of Vienna, Vienna, Austria.
  • Steudle F; Center for Brain Research, Medical University of Vienna, Vienna, Austria.
  • Puthenkalam R; Center for Brain Research, Medical University of Vienna, Vienna, Austria.
  • Ernst M; Center for Brain Research, Medical University of Vienna, Vienna, Austria petra.scholze@meduniwien.ac.at margot.ernst@meduniwien.ac.at.
  • Scholze P; Center for Brain Research, Medical University of Vienna, Vienna, Austria petra.scholze@meduniwien.ac.at margot.ernst@meduniwien.ac.at.
Mol Pharmacol ; 99(1): 39-48, 2021 01.
Article em En | MEDLINE | ID: mdl-33268553

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Benzodiazepinas / Receptores de GABA-A / Moduladores GABAérgicos Limite: Animals / Female / Humans Idioma: En Revista: Mol Pharmacol Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Áustria

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Benzodiazepinas / Receptores de GABA-A / Moduladores GABAérgicos Limite: Animals / Female / Humans Idioma: En Revista: Mol Pharmacol Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Áustria