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Monoacylglycerol lipase (MAGL) inhibitors based on a diphenylsulfide-benzoylpiperidine scaffold.
Bononi, Giulia; Tonarini, Giacomo; Poli, Giulio; Barravecchia, Ivana; Caligiuri, Isabella; Macchia, Marco; Rizzolio, Flavio; Demontis, Gian Carlo; Minutolo, Filippo; Granchi, Carlotta; Tuccinardi, Tiziano.
Afiliação
  • Bononi G; Department of Pharmacy, University of Pisa, Via Bonanno 6, 56126, Pisa, Italy.
  • Tonarini G; Department of Pharmacy, University of Pisa, Via Bonanno 6, 56126, Pisa, Italy.
  • Poli G; Department of Pharmacy, University of Pisa, Via Bonanno 6, 56126, Pisa, Italy.
  • Barravecchia I; Department of Pharmacy, University of Pisa, Via Bonanno 6, 56126, Pisa, Italy.
  • Caligiuri I; Pathology Unit, Centro di Riferimento Oncologico di Aviano (CRO) IRCCS, 33081, Aviano, Italy.
  • Macchia M; Department of Pharmacy, University of Pisa, Via Bonanno 6, 56126, Pisa, Italy.
  • Rizzolio F; Pathology Unit, Centro di Riferimento Oncologico di Aviano (CRO) IRCCS, 33081, Aviano, Italy; Department of Molecular Sciences and Nanosystems, Ca' Foscari University, 30123, Venezia, Italy.
  • Demontis GC; Department of Pharmacy, University of Pisa, Via Bonanno 6, 56126, Pisa, Italy.
  • Minutolo F; Department of Pharmacy, University of Pisa, Via Bonanno 6, 56126, Pisa, Italy; Center for Instrument Sharing of the University of Pisa (CISUP), Lungarno Pacinotti 43, 56126, Pisa, Italy.
  • Granchi C; Department of Pharmacy, University of Pisa, Via Bonanno 6, 56126, Pisa, Italy; Center for Instrument Sharing of the University of Pisa (CISUP), Lungarno Pacinotti 43, 56126, Pisa, Italy. Electronic address: carlotta.granchi@unipi.it.
  • Tuccinardi T; Department of Pharmacy, University of Pisa, Via Bonanno 6, 56126, Pisa, Italy; Center for Instrument Sharing of the University of Pisa (CISUP), Lungarno Pacinotti 43, 56126, Pisa, Italy.
Eur J Med Chem ; 223: 113679, 2021 Nov 05.
Article em En | MEDLINE | ID: mdl-34218085

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piperidinas / Sulfetos / Inibidores Enzimáticos / Monoacilglicerol Lipases Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Itália

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piperidinas / Sulfetos / Inibidores Enzimáticos / Monoacilglicerol Lipases Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Itália