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Synthesis of novel hybrid pharmacophore of N-((4-sulfamoylphenyl)carbamothioyl)alkanamides as potent carbonic anhydrase-II and 15-lipoxygenase inhibitors.
Saeed, Aamer; Khan, Shafi Ullah; Saeed, Maria; Shabir, Ghulam; Hasan, Abbas; Khera, Rasheed Ahmad; El-Seedi, Hesham; Halim, Sobia Ahsan; Khan, Ajmal; Al-Harrasi, Ahmed; Iqbal, Jamshed.
Afiliação
  • Saeed A; Department of Chemistry, Quaid-i-Azam University, Islamabad, Pakistan.
  • Khan SU; Centre for Advanced Drug Research, COMSATS Institute of Information Technology, Abbottabad, Pakistan.
  • Saeed M; Department of Pharmacy, Abasyn University, Peshawar, Pakistan.
  • Shabir G; Department of Chemistry, Quaid-i-Azam University, Islamabad, Pakistan.
  • Hasan A; Department of Chemistry, Quaid-i-Azam University, Islamabad, Pakistan.
  • Khera RA; Department of Chemistry, Quaid-i-Azam University, Islamabad, Pakistan.
  • El-Seedi H; Department of Chemistry, University of Agriculture, Faisalabad, Pakistan.
  • Halim SA; International Research Center for Food Nutrition and Safety, Jiangsu University, Zhenjiang, China.
  • Khan A; International Joint Research Laboratory of Intelligent Agriculture and Agri-products Processing, Jiangsu Education Department, Jiangsu University, China.
  • Al-Harrasi A; Natural and Medical Sciences Research Center, University of Nizwa, Nizwa, Oman.
  • Iqbal J; Natural and Medical Sciences Research Center, University of Nizwa, Nizwa, Oman.
Drug Dev Res ; 83(3): 745-754, 2022 05.
Article em En | MEDLINE | ID: mdl-34897776

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Inibidores de Lipoxigenase / Anidrase Carbônica II Limite: Animals Idioma: En Revista: Drug Dev Res Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Paquistão

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Inibidores de Lipoxigenase / Anidrase Carbônica II Limite: Animals Idioma: En Revista: Drug Dev Res Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Paquistão