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Filarial nematode phenotypic screening cascade to identify compounds with anti-parasitic activity for drug discovery optimization.
Hawryluk, Natalie; Zhiru, Li; Carlow, Clotilde; Gokool, Suzanne; Townson, Simon; Kreiss, Tamara; Chojnowski, Agnieszka; Prorok, Monika; Siekierka, John; Ehrens, Alexandra; Koschel, Marianne; Lhermitte-Vallarino, Nathaly; Martin, Coralie; Hoerauf, Achim; Hernandez, Geraldine; Canan, Stacie; Khetani, Vikram; Zeldis, Jerome; Specht, Sabine; Hübner, Marc P; Scandale, Ivan.
Afiliação
  • Hawryluk N; Bristol Myers Squibb, San Diego, CA, USA. Electronic address: nataliehawryluk@gmail.com.
  • Zhiru L; New England Biolabs, Ipswich, MA, USA.
  • Carlow C; New England Biolabs, Ipswich, MA, USA.
  • Gokool S; Northwick Park Institute for Medical Research, London, UK.
  • Townson S; Northwick Park Institute for Medical Research, London, UK.
  • Kreiss T; Sokol Institute of Pharmaceutical Life Sciences, Montclair State University, Montclair, NJ, USA.
  • Chojnowski A; Sokol Institute of Pharmaceutical Life Sciences, Montclair State University, Montclair, NJ, USA.
  • Prorok M; Sokol Institute of Pharmaceutical Life Sciences, Montclair State University, Montclair, NJ, USA.
  • Siekierka J; Sokol Institute of Pharmaceutical Life Sciences, Montclair State University, Montclair, NJ, USA.
  • Ehrens A; Institute for Medical Microbiology, Immunology and Parasitology, University Hospital Bonn, Germany; German Center for Infection Research (DZIF), Partner Site Bonn-Cologne, Bonn, Germany.
  • Koschel M; Institute for Medical Microbiology, Immunology and Parasitology, University Hospital Bonn, Germany.
  • Lhermitte-Vallarino N; German Center for Infection Research (DZIF), Partner Site Bonn-Cologne, Bonn, Germany.
  • Martin C; Unité Molécules de Communication et Adaptation des Microorganismes (MCAM, UMR 7245), Muséum national d'Histoire naturelle, Paris, France.
  • Hoerauf A; Institute for Medical Microbiology, Immunology and Parasitology, University Hospital Bonn, Germany; German Center for Infection Research (DZIF), Partner Site Bonn-Cologne, Bonn, Germany.
  • Hernandez G; Bristol Myers Squibb, San Diego, CA, USA.
  • Canan S; Bristol Myers Squibb, San Diego, CA, USA.
  • Khetani V; Bristol Myers Squibb, Summit, NJ, USA.
  • Zeldis J; Celgene Global Health, Summit, NJ, USA.
  • Specht S; Institute for Medical Microbiology, Immunology and Parasitology, University Hospital Bonn, Germany; Drugs for Neglected Diseases Initiative, Geneva, Switzerland.
  • Hübner MP; Institute for Medical Microbiology, Immunology and Parasitology, University Hospital Bonn, Germany; German Center for Infection Research (DZIF), Partner Site Bonn-Cologne, Bonn, Germany.
  • Scandale I; Drugs for Neglected Diseases Initiative, Geneva, Switzerland.
Article em En | MEDLINE | ID: mdl-35834918

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Oncocercose / Parasitos / Brugia Malayi Tipo de estudo: Diagnostic_studies / Screening_studies Limite: Adult / Animals / Humans Idioma: En Revista: Int J Parasitol Drugs Drug Resist Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Oncocercose / Parasitos / Brugia Malayi Tipo de estudo: Diagnostic_studies / Screening_studies Limite: Adult / Animals / Humans Idioma: En Revista: Int J Parasitol Drugs Drug Resist Ano de publicação: 2022 Tipo de documento: Article