Discovery and Mechanistic Analysis of Structurally Diverse Inhibitors of Acetyltransferase Eis among FDA-Approved Drugs.

Pang, Allan H; Green, Keith D; Punetha, Ankita; Thamban Chandrika, Nishad; Howard, Kaitlind C; Garneau-Tsodikova, Sylvie; Tsodikov, Oleg V

Pang, Allan H; Green, Keith D; Punetha, Ankita; Thamban Chandrika, Nishad; Howard, Kaitlind C; Garneau-Tsodikova, Sylvie; Tsodikov, Oleg V.

Afiliação

Pang AH; Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, 789 South Limestone Street, Lexington, Kentucky40536-0596, United States.
Green KD; Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, 789 South Limestone Street, Lexington, Kentucky40536-0596, United States.
Punetha A; Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, 789 South Limestone Street, Lexington, Kentucky40536-0596, United States.
Thamban Chandrika N; Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, 789 South Limestone Street, Lexington, Kentucky40536-0596, United States.
Howard KC; Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, 789 South Limestone Street, Lexington, Kentucky40536-0596, United States.
Garneau-Tsodikova S; Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, 789 South Limestone Street, Lexington, Kentucky40536-0596, United States.
Tsodikov OV; Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, 789 South Limestone Street, Lexington, Kentucky40536-0596, United States.

Biochemistry ; 62(3): 710-721, 2023 02 07.

Article em En | MEDLINE | ID: mdl-36657084

Assuntos

Acetiltransferases; Mycobacterium tuberculosis; Tuberculose; Humanos; Acetiltransferases/antagonistas & inibidores; Antituberculosos/farmacologia; Antituberculosos/química; Proteínas de Bactérias/antagonistas & inibidores; Canamicina/farmacologia; Canamicina/química; Mycobacterium tuberculosis/efeitos dos fármacos; Mycobacterium tuberculosis/enzimologia; Proguanil/metabolismo; Tuberculose/tratamento farmacológico

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Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Acetiltransferases / Tuberculose / Mycobacterium tuberculosis Limite: Humans Idioma: En Revista: Biochemistry Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Estados Unidos

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