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Paralog-dependent isogenic cell assay cascade generates highly selective SLC16A3 inhibitors.
Dvorak, Vojtech; Casiraghi, Andrea; Colas, Claire; Koren, Anna; Tomek, Tatjana; Offensperger, Fabian; Rukavina, Andrea; Tin, Gary; Hahn, Elisa; Dobner, Sarah; Frommelt, Fabian; Boeszoermenyi, Andras; Bernada, Viktoriia; Hannich, J Thomas; Ecker, Gerhard F; Winter, Georg E; Kubicek, Stefan; Superti-Furga, Giulio.
Afiliação
  • Dvorak V; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Casiraghi A; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Colas C; Department of Pharmaceutical Sciences, University of Vienna, 1090 Vienna, Austria.
  • Koren A; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Tomek T; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Offensperger F; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Rukavina A; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Tin G; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Hahn E; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Dobner S; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Frommelt F; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Boeszoermenyi A; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Bernada V; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Hannich JT; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Ecker GF; Department of Pharmaceutical Sciences, University of Vienna, 1090 Vienna, Austria.
  • Winter GE; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Kubicek S; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.
  • Superti-Furga G; CeMM Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria; Center for Physiology and Pharmacology, Medical University of Vienna, 1090 Vienna, Austria. Electronic address: GSuperti@cemm.oeaw.ac.at.
Cell Chem Biol ; 30(8): 953-964.e9, 2023 08 17.
Article em En | MEDLINE | ID: mdl-37516113

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Proteínas de Transporte / Descoberta de Drogas Tipo de estudo: Prognostic_studies Idioma: En Revista: Cell Chem Biol Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Áustria

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Proteínas de Transporte / Descoberta de Drogas Tipo de estudo: Prognostic_studies Idioma: En Revista: Cell Chem Biol Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Áustria