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Discovery of Biaryl Amide Derivatives as Potent, Selective, and Orally Bioavailable RORγt Agonists for Cancer Immunotherapy.
Lu, Lixue; Huang, Yafei; Song, Meiqi; Sun, Nannan; Xia, Li; Yu, Mingcheng; Zhao, Meiling; Qiu, Ruomeng; Chen, Ji-An; Zhao, Yunpeng; Wang, Haojie; Guo, Huimin; Li, Yan; Zhu, Di; Wang, Yonghui; Xie, Qiong.
Afiliação
  • Lu L; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Huang Y; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Song M; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Sun N; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Xia L; School of Pharmaceutical Sciences, Zhengzhou University, Zhengzhou 450001, China.
  • Yu M; Department of Pharmacology, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Zhao M; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Qiu R; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Chen JA; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Zhao Y; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Wang H; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Guo H; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Li Y; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Zhu D; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Wang Y; Department of Pharmacology, School of Pharmacy, Fudan University, Shanghai 201203, China.
  • Xie Q; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
J Med Chem ; 66(23): 16091-16108, 2023 12 14.
Article em En | MEDLINE | ID: mdl-37982494

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Amidas / Neoplasias Limite: Animals Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: China

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Amidas / Neoplasias Limite: Animals Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: China